SCHEMBL20839781

SCHEMBL20839781

Cc1ccc(NC(=O)c2ccc3ccccc3c2)c(C(=O)Nc2cccc(CCC(=O)O)c2)c1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 11/20 0.71
PPARD Q03181 7/20 0.70
PPARG P37231 7/20 0.64
PPARA Q07869 5/20 0.64
F10 P00742 1/20 0.63
HSPH1 Q92598 1/20 0.58
ITGB3 P05106 1/20 0.52
ITGA2B P08514 1/20 0.52
RXFP1 Q9HBX9 1/20 0.50
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20839737 0.92 NR1H4 (0.80) NR1H4PPARDPPARGPPARAF10
SCHEMBL20839645 0.90 NR1H4 (0.73) NR1H4PPARDPPARGPPARAF10
SCHEMBL20839783 0.89 NR1H4 (0.80) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20840618 0.89 NR1H4 (0.59) NR1H4PPARDPPARGPPARAF10
SCHEMBL20839666 0.89 NR1H4 (0.86) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839667 0.89 HSPH1 (0.73) NR1H4PPARDPPARGPPARAF10
SCHEMBL6594035 0.85 F10 (0.83) NR1H4PPARDPPARGPPARAF10
SCHEMBL20839624 0.85 NR1H4 (0.78) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20852075 0.84 NR1H4 (0.68) NR1H4PPARDPPARGPPARAHSPH1
SCHEMBL20839500 0.83 NR1H4 (1.00) NR1H4PPARDPPARGPPARAHSPH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed
WO-2019057969-A1 DUAL AGONISTS OF FXR AND PPARδ AND THEIR USES Johann Wolfgang Goethe-Universität (DE) 2019-03-28 WO disclosed