SCHEMBL20852503

SCHEMBL20852503

CCn1c(=O)c(-c2cc(NC(=O)Nc3ccc(F)cc3)c(F)cc2F)cc2cnc(NC)cc21

nearest known ligand 0.76

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KIT P10721 1/20 0.76
PDGFRA P16234 1/20 0.76
RAF1 P04049 4/20 0.63
BRAF P15056 4/20 0.63
KRAS P01116 3/20 0.63
KDR P35968 3/20 0.63
MAP2K2 P36507 3/20 0.63
MAP2K1 Q02750 3/20 0.63
BTK Q06187 12/20 0.51
SRC P12931 9/20 0.51
LYN P07948 7/20 0.51
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ARAF P10398 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15000252 0.94 KIT (0.86) KITPDGFRARAF1BRAFKRAS
SCHEMBL15006335 0.92 KIT (0.70) KITPDGFRARAF1BRAFKRAS
SCHEMBL15006336 0.92 KIT (0.72) KITPDGFRARAF1BRAFKRAS
SCHEMBL20852376 0.92 KIT (0.64) KITPDGFRARAF1BRAFKRAS
SCHEMBL29800429 0.92 KIT (0.64) KITPDGFRARAF1BRAFKRAS
Hydrochloric Acid SCHEMBL21796167 0.91 KIT (0.69) KITPDGFRARAF1BRAFKRAS
Hydrochloric Acid SCHEMBL21796184 0.91 KIT (0.71) KITPDGFRARAF1BRAFKRAS
SCHEMBL14999838 0.91 KIT (0.75) KITPDGFRARAF1BRAFKRAS
SCHEMBL17244719 0.89 KIT (0.68) KITPDGFRARAF1BRAFKRAS
SCHEMBL15000009 0.88 KIT (0.73) KITPDGFRARAF1BRAFKRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019056990-A1 1,2-DIHYDRO-1,6-NAPHTHYRIDINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN MEDICINE 浙江海正药业股份有限公司 2019-03-28 WO disclosed