SCHEMBL29800429

SCHEMBL29800429

CNc1cc2c(cn1)cc(-c1cc(NC(=O)Nc3ccc(F)cc3)c(F)cc1F)c(=O)n2CC(F)(F)F

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIT P10721 1/20 0.64
PDGFRA P16234 1/20 0.64
BRAF P15056 10/20 0.55
RAF1 P04049 9/20 0.55
KRAS P01116 6/20 0.55
KDR P35968 6/20 0.55
MAP2K2 P36507 5/20 0.55
MAP2K1 Q02750 5/20 0.55
SRC P12931 5/20 0.42
BTK Q06187 5/20 0.42
LYN P07948 4/20 0.42
ARAF P10398 2/20 0.41
FGFR1 P11362 1/20 0.39
FGFR4 P22455 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20852376 1.00 KIT (0.64) KITPDGFRABRAFRAF1KRAS
SCHEMBL20852395 0.94 BRAF (0.64) KITPDGFRABRAFRAF1KRAS
SCHEMBL29800826 0.94 BRAF (0.64) KITPDGFRABRAFRAF1KRAS
SCHEMBL20852503 0.92 KIT (0.76) KITPDGFRABRAFRAF1KRAS
SCHEMBL29800828 0.91 KIT (0.64) KITPDGFRABRAFRAF1KRAS
SCHEMBL20852384 0.91 KIT (0.64) KITPDGFRABRAFRAF1KRAS
SCHEMBL20852461 0.89 KIT (0.51) KITPDGFRABRAFRAF1KRAS
SCHEMBL20852397 0.86 KIT (0.86) KITPDGFRABRAFRAF1KRAS
SCHEMBL20852396 0.86 KIT (0.71) KITPDGFRABRAFRAF1KRAS
SCHEMBL29800851 0.86 KIT (0.86) KITPDGFRABRAFRAF1KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111094286-B 1, 2-dihydro-1, 6-naphthyridine derivatives, preparation method and medical application thereof 浙江海正药业股份有限公司 2022-07-29 CN disclosed