SCHEMBL20856476

SCHEMBL20856476

CCOc1ccc2c(N)c3ccc(N)cc3nc2c1

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.86
KMT2A Q03164 4/20 0.86
BLM P54132 2/20 0.86
TERT O14746 1/20 0.86
ABCB11 O95342 1/20 0.86
LMNA P02545 1/20 0.86
THRB P10828 1/20 0.86
CASP7 P55210 3/20 0.69
CASP1 P29466 2/20 0.69
ALDH1A1 P00352 2/20 0.69
HSD17B10 Q99714 2/20 0.69
KDM4E B2RXH2 1/20 0.69
MAPT P10636 1/20 0.69
HPGD P15428 1/20 0.69
MAPK1 P28482 1/20 0.69
ELANE P08246 1/20 0.52
APAF1 O14727 1/20 0.52
POLB P06746 1/20 0.52
CASP3 P42574 1/20 0.52
CASP6 P55212 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethacridine SCHEMBL193949 0.93 MEN1 (1.00) MEN1KMT2ABLMTERTABCB11
Ethacridine SCHEMBL30310148 0.93 MEN1 (1.00) MEN1KMT2ABLMTERTABCB11
Ethacridine SCHEMBL11662539 0.93 MEN1 (1.00) MEN1KMT2ABLMTERTABCB11
Ethacridine SCHEMBL29456272 0.93 MEN1 (1.00) MEN1KMT2ABLMTERTABCB11
Ethacridine SCHEMBL30753462 0.91 MEN1 (0.97) MEN1KMT2ABLMTERTABCB11
Ethacridine SCHEMBL9355974 0.91 MEN1 (0.97) MEN1KMT2ABLMTERTABCB11
Lactic Acid SCHEMBL8375854 0.87 MEN1 (0.91) MEN1KMT2ABLMTERTABCB11
Ethacridine SCHEMBL7041699 0.86 MEN1 (0.85) MEN1KMT2ABLMTERTABCB11
Ethacridine SCHEMBL31197660 0.83 MEN1 (1.00) MEN1KMT2ABLMTERTABCB11
Ethacridine SCHEMBL30006678 0.83 MEN1 (1.00) MEN1KMT2ABLMTERTABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12247246-B2 Identification of inhibitors of TcpC and TIR NADase activity WASHINGTON UNIVERSITY (US) 2025-03-11 US disclosed
US-20230272449-A1 IDENTIFICATION OF INHIBITORS OF TCPC AND TIR NADase ACTIVITY WASHINGTON UNIVERSITY 2023-08-31 US disclosed
US-20200283820-A1 IDENTIFICATION OF INHIBITORS OF TCPC AND TIR NADase ACTIVITY WASHINGTON UNIVERSITY 2020-09-10 US disclosed
WO-2019067625-A1 IDENTIFICATION OF INHIBITORS OF TCPC AND TIR NADASE ACTIVITY WASHINGTON UNIVERSITY (US) 2019-04-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230272449-A1 IDENTIFICATION OF INHIBITORS OF TCPC AND TIR NADase ACTIVITY NADK, NAPRT, TIPARP MEN1 3678/4885KMT2A 3095/4885BLM 2925/4885
US-12247246-B2 Identification of inhibitors of TcpC and TIR NADase activity NADK, NAPRT, TIPARP MEN1 3678/4885KMT2A 3095/4885BLM 2925/4885
US-20200283820-A1 IDENTIFICATION OF INHIBITORS OF TCPC AND TIR NADase ACTIVITY NADK, NAPRT, TIPARP MEN1 3678/4885KMT2A 3095/4885BLM 2925/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.