SCHEMBL20869211

SCHEMBL20869211

COc1ccc(C(F)(F)F)nc1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 12/20 0.48
KDM4E B2RXH2 3/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
PDE4A P27815 3/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
PDE3A Q14432 1/20 0.40
TGFBR1 P36897 1/20 0.40
CXCR4 P61073 1/20 0.40
HPGD P15428 2/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PTGS2 P35354 3/20 0.39
PTGS1 P23219 2/20 0.39
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31010990 0.78 PDE4B (0.45) PDE4BKDM4EPDE4APDE4CPDE4D
SCHEMBL18606101 0.78 PDE4B (0.45) PDE4BKDM4EPDE4APDE4CPDE4D
SCHEMBL30358862 0.78 PDE4B (0.43) PDE4BKDM4EPDE4APDE4CPDE4D
SCHEMBL7917474 0.78 PDE4B (0.43) PDE4BKDM4EPDE4APDE4CPDE4D
SCHEMBL12062521 0.78 KDM4E (0.49) KDM4EL3MBTL1TGFBR1SMN1; SMN2ALDH1A1
SCHEMBL25601599 0.78 PDE4B (0.39) PDE4BKDM4EPDE4APDE4CPDE4D
SCHEMBL12538667 0.78 TRPV3 (0.56) HPGDLMNATP53HTTKMT2A
SCHEMBL25791611 0.77 PDE4B (0.43) PDE4BKDM4EL3MBTL1PDE4APDE4C
SCHEMBL23554835 0.76 PDE4B (0.52) PDE4BPDE4APDE4CPDE4DPDE3A
SCHEMBL29550138 0.76 PDE4B (0.52) PDE4BPDE4APDE4CPDE4DPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019063748-A1 ROR-GAMMA INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-04-04 WO disclosed
CN-104254525-B aromatic ring compound TAKEDA PHARMACEUTICAL CO.,LTD. (JP) 2016-05-25 CN disclosed
CN-104254525-A Aromatic ring compound TAKEDA PHARMACEUTICAL 2014-12-31 CN disclosed
CN-101677569-B 2-cyanophenyl fused heterocyclic compounds, and compositions and uses thereof EVOTEC AG 2014-01-22 CN disclosed
CN-101677569-A 2-cyanophenyl fused heterocyclic compounds, and compositions and uses thereof RENOVIS INC 2010-03-24 CN disclosed