SCHEMBL20909052

SCHEMBL20909052

C[C@H]1CC2(CCN(c3ncc(-c4cc5ccccc5n4C)nc3CO)CC2)CO1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 16/20 0.42
CYP11B2 P19099 2/20 0.39
TRPV3 Q8NET8 1/20 0.34
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22594931 0.89 PTPN11 (0.39) PTPN11CYP11B2TRPV3KCNH2
SCHEMBL20909038 0.85 CYP11B2 (0.45) PTPN11CYP11B2TRPV3
SCHEMBL30787853 0.83 PTPN11 (0.63) PTPN11KCNH2
SCHEMBL20899399 0.83 PTPN11 (0.63) PTPN11KCNH2
SCHEMBL20909039 0.78 PTPN11 (0.47) PTPN11KCNH2
SCHEMBL22594980 0.77 PTPN11 (0.50) PTPN11
SCHEMBL20909056 0.77 PTPN11 (0.68) PTPN11KCNH2
SCHEMBL22594735 0.77 PTPN11 (0.62) PTPN11
SCHEMBL20909050 0.77 PTPN11 (0.69) PTPN11KCNH2
SCHEMBL24151104 0.76 PTPN11 (0.42) PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019075265-A1 PYRIDINE, PYRAZINE, AND TRIAZINE COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS Revolution Medicines, Inc. (US) 2019-04-18 WO disclosed