SCHEMBL20912425

SCHEMBL20912425

COc1ccc2c(c1)C(=N)c1nc3ncccc3c(=O)n1-2

nearest known ligand 0.79

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 17/20 0.79
PDE10A Q9Y233 1/20 0.45
MMP10 P09238 1/20 0.44
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5619918 0.88 IDO1 (1.00) IDO1PDE10A
SCHEMBL19456573 0.86 IDO1 (0.77) IDO1
SCHEMBL20912427 0.86 IDO1 (0.80) IDO1
SCHEMBL20597738 0.84 IDO1 (0.74) IDO1PDE10A
SCHEMBL30141739 0.84 IDO1 (0.74) IDO1PDE10A
SCHEMBL19456481 0.84 IDO1 (0.74) IDO1PDE10A
SCHEMBL20912413 0.82 IDO1 (0.78) IDO1
SCHEMBL19456420 0.82 IDO1 (0.78) IDO1
SCHEMBL19456589 0.82 IDO1 (0.72) IDO1PDE10A
SCHEMBL19456513 0.80 IDO1 (0.75) IDO1LMNAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10669273-B2 Use of aza-tryptanthrin derivatives as inhibitors of IDO1 and/or TDO PEKING UNIVERSITY (CN) 2020-06-02 US disclosed
US-20190112308-A1 Use of Aza-Tryptanthrin Derivatives as Inhibitors of IDO1 and/or TDO PEKING UNIVERSITY (CN) 2019-04-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10669273-B2 Use of aza-tryptanthrin derivatives as inhibitors of IDO1 and/or TDO IDO1, TDO2, IDO2 IDO1 1/4885PDE10A 3741/4885MMP10 1665/4885
US-20190112308-A1 Use of Aza-Tryptanthrin Derivatives as Inhibitors of IDO1 and/or TDO IDO1, TDO2, IDO2 IDO1 1/4885PDE10A 3741/4885MMP10 1665/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.