SCHEMBL20913056

SCHEMBL20913056

COC(=O)/C=C/C1=C(OS(=O)(=O)C(F)(F)F)CCN(C(=O)O)C1C

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.33
DRD3 P35462 5/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19874445 1.00 DRD2 (0.33) DRD2DRD3
SCHEMBL19874349 0.89 NR1H2 (0.33) DRD2DRD3
SCHEMBL19886463 0.78 NR1H2 (0.32)
SCHEMBL19874448 0.76 GPER1 (0.32) DRD2DRD3
SCHEMBL19874447 0.76 GPER1 (0.32) DRD2DRD3
SCHEMBL19874403 0.75 DRD2 (0.33) DRD2DRD3
SCHEMBL19874400 0.75 DRD2 (0.33) DRD2DRD3
SCHEMBL19874372 0.69 NR1H2 (0.36) DRD2DRD3
SCHEMBL19874374 0.69 NR1H2 (0.36) DRD2DRD3
SCHEMBL19874306 0.68 GPER1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3265465-B1 BICYCLIC KETONE SULFONAMIDE COMPOUNDS AMGEN INC (US) 2019-04-24 EP disclosed