SCHEMBL20935192

SCHEMBL20935192

C=CC1(F)CN(C(=O)OC(C)(C)C)CCC1Oc1cnc(-c2ccnc(Nc3ccc(N4CCN(C5COC5)CC4)c(OC)n3)n2)cc1C#N

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 19/20 0.46
IKBKE Q14164 2/20 0.46
JAK2 O60674 13/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24904172 0.93 TBK1 (0.52) TBK1IKBKEJAK2
SCHEMBL20934839 0.86 TBK1 (0.59) TBK1IKBKEJAK2
SCHEMBL20935193 0.85 TBK1 (0.46) TBK1IKBKEJAK2
SCHEMBL24904182 0.85 TBK1 (0.51) TBK1IKBKEJAK2
SCHEMBL20935203 0.84 TBK1 (0.63) TBK1IKBKEJAK2
SCHEMBL20935204 0.84 TBK1 (0.63) TBK1IKBKEJAK2
SCHEMBL20934764 0.84 TBK1 (0.49) TBK1IKBKEJAK2
SCHEMBL24904181 0.83 TBK1 (0.52) TBK1IKBKEJAK2
SCHEMBL20935147 0.81 TBK1 (0.67) TBK1IKBKEJAK2
SCHEMBL24904170 0.81 TBK1 (0.56) TBK1IKBKEJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019079373-A1 PYRIMIDINE TBK/IKKε INHIBITOR COMPOUNDS AND USES THEREOF MERCK PATENT GMBH (DE) 2019-04-25 WO disclosed