SCHEMBL20976589

SCHEMBL20976589

COC1COCCC1NC1CCN(C(=O)c2nc(C3CCOCC3)nc(N3CCc4ccc(C(F)(F)F)cc4C3)c2C)CC1

nearest known ligand 0.80

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 19/20 0.80
CCR5 P51681 3/20 0.80
KCNH2 Q12809 3/20 0.53
CCR1 P32246 1/20 0.44
TMEM97 Q5BJF2 1/20 0.44
SIGMAR1 Q99720 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15081517 1.00 CCR2 (0.80) CCR2CCR5KCNH2CCR1TMEM97
SCHEMBL15081515 1.00 CCR2 (0.80) CCR2CCR5KCNH2CCR1TMEM97
SCHEMBL14945898 0.98 CCR2 (0.81) CCR2CCR5KCNH2CCR1TMEM97
SCHEMBL14945902 0.98 CCR2 (0.81) CCR2CCR5KCNH2CCR1TMEM97
SCHEMBL15081508 0.97 CCR2 (0.84) CCR2CCR5KCNH2CCR1TMEM97
SCHEMBL20976586 0.97 CCR2 (0.84) CCR2CCR5KCNH2CCR1TMEM97
SCHEMBL15081475 0.97 CCR2 (0.84) CCR2CCR5KCNH2CCR1TMEM97
SCHEMBL20976601 0.95 CCR2 (0.73) CCR2CCR5KCNH2CCR1TMEM97
SCHEMBL20976575 0.91 CCR2 (0.95) CCR2CCR5KCNH2CCR1TMEM97
SCHEMBL15081425 0.91 CCR2 (0.66) CCR2CCR5KCNH2TMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2731941-B1 NOVEL AND SELECTIVE CCR2 ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2019-05-08 EP disclosed