SCHEMBL20979520

SCHEMBL20979520

C/C(=N\NC(=O)c1cccc([S+]([O-])N2CCOCC2)c1)c1cccc(Cl)c1F

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.49
BRD4 O60885 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
BRD2 P25440 1/20 0.48
CYP2C19 P33261 1/20 0.48
MTOR P42345 3/20 0.47
MAPT P10636 6/20 0.45
NPC1 O15118 2/20 0.44
ALDH1A1 P00352 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.41
GAA P10253 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22213034 0.88 KDM1A (0.57) KDM1ABRD4CYP3A4CYP2C9BRD2
SCHEMBL20979639 0.86 KDM1A (0.58) KDM1ABRD4CYP3A4CYP2C9BRD2
SCHEMBL20979524 0.84 KDM1A (0.70) KDM1ABRD4CYP3A4CYP2C9BRD2
SCHEMBL20979632 0.82 KDM1A (0.50) KDM1ABRD4CYP3A4CYP2C9BRD2
SCHEMBL20979562 0.80 MAPT (0.47) KDM1ABRD4CYP3A4CYP2C9BRD2
SCHEMBL15772600 0.80 KDM1A (0.75) KDM1ABRD4CYP3A4CYP2C9BRD2
SCHEMBL14712680 0.80 KDM1A (0.75) KDM1ABRD4CYP3A4CYP2C9BRD2
SCHEMBL15772602 0.80 KDM1A (0.75) KDM1ABRD4CYP3A4CYP2C9BRD2
SCHEMBL22213030 0.79 RAB9A (0.54) MTORMAPTNPC1ALDH1A1SMN1; SMN2
SCHEMBL22213035 0.76 KDM1A (0.56) KDM1ABRD4CYP3A4CYP2C9BRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3010915-B1 SUBSTITUTED (3-(5-CHLORO-2-HYDROXYPHENYL)-1-BENZOYL-1H-PYRAZOLE COMPOUNDS AS HISTONE DEMETHYLASE INHIBITORS UNIV UTAH RES FOUND (US) 2019-05-08 EP disclosed