SCHEMBL209885

SCHEMBL209885

N[C@@H](CCCCN(Cc1ccccc1)Cc1ccccc1)C(=O)O

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP7 Q9UHL4 2/20 0.66
DPP8 Q6V1X1 1/20 0.66
DPP9 Q86TI2 1/20 0.66
HDAC3 O15379 2/20 0.54
HDAC1 Q13547 2/20 0.54
HDAC2 Q92769 2/20 0.54
HDAC8 Q9BY41 2/20 0.54
NCOR2 Q9Y618 2/20 0.54
POLB P06746 1/20 0.52
KMT2A Q03164 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
ALPI P09923 1/20 0.50
PKM P14618 1/20 0.50
PTGS1 P23219 1/20 0.50
XIAP P98170 1/20 0.50
SLC7A5 Q01650 1/20 0.50
GRIK1 P39086 1/20 0.47
SLC1A5 Q15758 7/20 0.46
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7044835 0.85 BCHE (0.53) DPP7DPP8DPP9POLBKMT2A
SCHEMBL209926 0.85 SIGMAR1 (0.54) DPP7DPP8DPP9POLBKMT2A
SCHEMBL21054744 0.85 SIGMAR1 (0.54) DPP7DPP8DPP9POLBKMT2A
SCHEMBL23656532 0.82 FOLH1 (0.60) DPP7DPP8DPP9POLBKMT2A
SCHEMBL27462545 0.82 LPAR1 (0.49) DPP7DPP8DPP9HDAC3HDAC1
SCHEMBL6172479 0.81 DPP7 (0.76) DPP7DPP8DPP9HDAC3HDAC1
SCHEMBL12977607 0.80 SLC1A5 (0.60) DPP7DPP8DPP9HDAC3HDAC1
SCHEMBL996075 0.80 SLC1A5 (0.60) DPP7DPP8DPP9HDAC3HDAC1
Hydrochloric Acid SCHEMBL7043275 0.79 KDM4A (0.50) DPP7DPP8DPP9KMT2AALPI
SCHEMBL2237757 0.79 SLC1A5 (0.47) DPP7DPP8DPP9POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1290 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1163262-B1 PHENYLALANINE DERIVATIVES US GOV HEALTH & HUMAN SERV (US) 2011-05-11 EP claimed
US-20080139456-A1 Macrocyclic Sh2 Domain Binding Inhibitors GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES 2008-06-12 US claimed
WO-2008067270-A1 MACROCYCLIC GRB2 SH2 DOMAIN-BINDING INHIBITORS GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2008-06-05 WO claimed
EP-1793843-A1 MACROCYCLIC SH2 DOMAIN BINDING INHIBITORS Government of the United States of America, Represented by the Secretary, Department of Health and Human Services (US) 2007-06-13 EP claimed
US-7226991-B1 inhibiting SH2 domain binding with a phosphoprotein; to inhibit proliferation of tumor cells; for inhibiting the growth of human breast cancer cells UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2007-06-05 US claimed
WO-2006039527-A1 MACROCYCLIC SH2 DOMAIN BINDING INHIBITORS GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2006-04-13 WO claimed
US-6977241-B2 SH2 domain binding inhibitors THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2005-12-20 US claimed
US-20040048788-A1 Sh2 domain binding inhibitors DEPARTMENT OF HEALTH AND HUMAN SERVICES, UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY, OF THE 2004-03-11 US claimed
EP-1383792-A2 SH2 DOMAIN BINDING INHIBITORS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2004-01-28 EP claimed
WO-2004003005-A2 SH2 DOMAIN BINDING INHIBITORS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2004-01-08 WO claimed
WO-2002016407-A2 SH2 DOMAIN BINDING INHIBITORS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2002-02-28 WO claimed
EP-1163262-A1 PHENYLALANINE DERIVATIVES THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by THE SECRETARY of the DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2001-12-19 EP claimed
WO-2000056760-A1 PHENYLALANINE DERIVATIVES THE UNITED STATES OF AMERICA, REPRESENTED BY SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-09-28 WO claimed
WO-1997007131-A1 ACYLATED OLIGOPEPTIDES CONTAINING PHOSPHOTYROSINE AS INHIBITORS OF PROTEIN TYROSINE KINASES NOVARTIS AG (CH) 1997-02-27 WO claimed
US-20260146073-A1 T CELL RECEPTORS TARGETING MUTATED CDKN2A THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVIC (US) 2026-05-28 US disclosed
EP-4748856-A2 COMPOSITIONS AND METHODS FOR TREATING CANCER WITH SELF-DRIVING CHIMERIC ANTIGEN RECEPTORS Lentigen Technology, Inc. (US) 2026-05-27 EP disclosed
EP-4747362-A2 METHODS FOR RAPID MANUFACTURE OF ENGINEERED T CELLS EXPRESSING CHIMERIC ANTIGEN RECEPTORS Kyverna Therapeutics, Inc. (US) 2026-05-27 EP disclosed
US-6307090-B1 OXALYL ENDCAPPED; CONTAINING A BIVALENT RADICAL OF PHOSPHOTYROSINE OR A PHOSPHOTYROSINE MIMETIC THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2001-10-23 US disclosed
WO-2000056760-A1 PHENYLALANINE DERIVATIVES THE UNITED STATES OF AMERICA, REPRESENTED BY SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-09-28 WO disclosed
WO-1997007131-A1 ACYLATED OLIGOPEPTIDES CONTAINING PHOSPHOTYROSINE AS INHIBITORS OF PROTEIN TYROSINE KINASES NOVARTIS AG (CH) 1997-02-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260146073-A1 T CELL RECEPTORS TARGETING MUTATED CDKN2A TP53, CD74, HLA-C DPP7 3994/4885DPP8 3317/4885DPP9 3267/4885
US-20080139456-A1 Macrocyclic Sh2 Domain Binding Inhibitors ACP1, PPM1D, LASP1 DPP7 1369/4885DPP8 1610/4885DPP9 1626/4885
US-20040048788-A1 Sh2 domain binding inhibitors ACP1, PHLPP1, SORBS1 DPP7 2408/4885DPP8 2565/4885DPP9 2151/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.