SCHEMBL20994591

SCHEMBL20994591

Sc1nc(-c2ccccc2)nn1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
NR1H2 P55055 1/20 0.43
NR1H3 Q13133 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.41
PTGS1 P23219 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
KDM4A O75164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2339443 0.78 SMN1; SMN2 (0.59) NPC1RAB9ANR1H2NR1H3SMN1; SMN2
SCHEMBL2211208 0.78 SMN1; SMN2 (0.37) NPC1RAB9ASMN1; SMN2KDM4A
SCHEMBL21471362 0.77 KDM4A (0.47) NPC1RAB9ANR1H2NR1H3SMN1; SMN2
SCHEMBL14007393 0.77 NPC1 (0.52) NPC1RAB9ANR1H2NR1H3SMN1; SMN2
SCHEMBL13936045 0.76 SMN1; SMN2 (0.56) NPC1RAB9ANR1H2NR1H3SMN1; SMN2
SCHEMBL13936046 0.76 SMN1; SMN2 (0.56) NPC1RAB9ANR1H2NR1H3SMN1; SMN2
SCHEMBL10401729 0.74 SMN1; SMN2 (0.43) NPC1RAB9ASMN1; SMN2KDM4A
SCHEMBL11333361 0.74 NR1H3 (0.63) NPC1RAB9ANR1H2NR1H3SMN1; SMN2
SCHEMBL10361051 0.74 KDM4A (0.41) SMN1; SMN2KDM4A
SCHEMBL13921714 0.74 NR1H3 (0.58) NPC1RAB9ANR1H2NR1H3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2850068-B1 N-(phenyl)-2-[[3-(phenyl)-1H-1,2,4-triazol-5-yl]thio]-acetamide derivatives and related compounds as G protein coupled receptor 17 (GPCR17) modulators for use in the treatment of neuro-degenerative diseases UNIV DEGLI STUDI MILANO (IT) 2019-05-29 EP disclosed