SCHEMBL21023240

SCHEMBL21023240

CC(C)(C)C(=O)NCCC(=O)N1CCC(=C2C3=C(C=C=C=C3)C=Cc3ccccc32)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.37
MGLL Q99685 1/20 0.37
ABHD6 Q9BV23 1/20 0.37
SETD7 Q8WTS6 3/20 0.36
DRD2 P14416 4/20 0.36
HTR1A P08908 2/20 0.36
ABCB11 O95342 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
ADRA2A P08913 1/20 0.36
CYP2D6 P10635 1/20 0.36
CHRM1 P11229 1/20 0.36
TSHR P16473 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
CHRM3 P20309 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2867635 0.88 SETD7 (0.47) FAAHMGLLABHD6SETD7DRD2
SCHEMBL4874727 0.77 SETD7 (0.49) FAAHMGLLABHD6SETD7DRD2
SCHEMBL2861222 0.75 SIGMAR1 (0.53) FAAHMGLLABHD6SETD7DRD2
SCHEMBL12854661 0.74 SETD7 (0.48) FAAHMGLLABHD6SETD7DRD2
Hydrochloric Acid SCHEMBL2864381 0.74 KMT2A (0.49) FAAHMGLLABHD6SETD7DRD2
SCHEMBL2864116 0.73 SETD7 (0.42) FAAHMGLLABHD6SETD7DRD2
SCHEMBL12854640 0.73 SETD7 (0.42) FAAHMGLLABHD6SETD7DRD2
SCHEMBL4875045 0.73 SETD7 (0.42) FAAHMGLLABHD6SETD7DRD2
SCHEMBL4897050 0.72 SETD7 (0.43) FAAHMGLLABHD6SETD7DRD2
SCHEMBL2868342 0.71 SETD7 (0.49) FAAHMGLLABHD6SETD7DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3485881-A1 PERMANENTLY CHARGED SODIUM AND CALCIUM CHANNEL BLOCKERS AS ANTI-INFLAMMATORY AGENTS President and Fellows of Harvard College (US) 2019-05-22 EP disclosed