SCHEMBL21024973

SCHEMBL21024973

CCCC(C)(C)Cc1cnccn1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP19A1 P11511 1/20 0.33
BRS3 P32247 1/20 0.32
CYP3A4 P08684 2/20 0.31
HRH1 P35367 1/20 0.31
TDP1 Q9NUW8 1/20 0.30
KDM4E B2RXH2 2/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
CYP1A2 P05177 1/20 0.30
HSP90AA1 P07900 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23138108 0.85 CYP2D6 (0.33) CYP2D6CYP2C9CYP2C19CYP19A1CYP3A4
SCHEMBL19605073 0.82 CYP2D6 (0.31) CYP2D6CYP2C9CYP2C19CYP19A1BRS3
SCHEMBL1912682 0.78 HDAC3 (0.38) CYP2D6CYP2C9CYP2C19CYP3A4HRH1
SCHEMBL19465295 0.74 CYP1A2 (0.46) HRH1TDP1CYP1A2ALDH1A1
SCHEMBL11260406 0.74 CYP1A2 (0.31) CYP2D6CYP2C9CYP2C19CYP3A4KDM4E
SCHEMBL21025398 0.74 BRS3 (0.37) CYP2D6CYP2C9CYP2C19BRS3CYP3A4
SCHEMBL21025553 0.74 KDM4E (0.38) CYP2D6CYP2C9CYP2C19CYP19A1TDP1
SCHEMBL2021219 0.72 KDM4E (0.34) CYP2D6CYP2C9CYP2C19CYP19A1CYP3A4
SCHEMBL18647608 0.71 CYP1A2 (0.30) CYP2C9CYP2C19CYP3A4CYP1A2
SCHEMBL309452 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230041563-A1 N-(1,3,4-OXADIAZOL-2-YL)ARYLCARBOXAMIDES OR SALTS THEREOF, PREPARATION METHODS, HERBICIDAL COMPOSITIONS AND USES THEREOF QINGDAO KINGAGROOT CHEMICAL COMPOUND CO., LTD. (CN) 2023-02-09 US disclosed
US-10669252-B2 Benzazepine derivative, preparation method, pharmaceutical composition and use thereof Shanghai De Novo Pharmatech Co., Ltd. (CN) 2020-06-02 US disclosed
US-20190152941-A1 BENZAZEPINE DERIVATIVE, PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE THEREOF Shanghai De Novo Pharmatech Co., Ltd. (CN) 2019-05-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230041563-A1 N-(1,3,4-OXADIAZOL-2-YL)ARYLCARBOXAMIDES OR SALTS THEREOF, PREPARATION METHODS, HERBICIDAL COMPOSITIONS AND USES THEREOF CYP2B6, CBR3, CYP2A6 CYP2D6 4/4885CYP2C9 48/4885CYP2C19 235/4885
US-10669252-B2 Benzazepine derivative, preparation method, pharmaceutical composition and use thereof TLR8, TLR1, TLR5 CYP2D6 894/4885CYP2C9 373/4885CYP2C19 317/4885
US-20190152941-A1 BENZAZEPINE DERIVATIVE, PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USE THEREOF TLR8, TLR1, TLR5 CYP2D6 894/4885CYP2C9 373/4885CYP2C19 317/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.