SCHEMBL21031949

SCHEMBL21031949

Cc1c(-c2csc3cc(-c4ccncc4)ccc23)c2cc(F)ccc2n1CC(=O)O

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 20/20 0.52
CYP2C9 P11712 1/20 0.48
PTGDR Q13258 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21032556 0.89 PTGDR2 (0.53) PTGDR2CYP2C9PTGDR
SCHEMBL21032707 0.87 MAPK14 (0.43) PTGDR2
SCHEMBL24180030 0.87 PTGDR2 (0.50) PTGDR2CYP2C9PTGDR
SCHEMBL21032554 0.86 PTGDR2 (0.49) PTGDR2CYP2C9PTGDR
SCHEMBL21032561 0.84 PTGDR2 (0.59) PTGDR2CYP2C9PTGDR
SCHEMBL24179951 0.84 PTGDR2 (0.56) PTGDR2CYP2C9PTGDR
SCHEMBL21032469 0.83 PTGDR2 (0.60) PTGDR2CYP2C9PTGDR
SCHEMBL21032885 0.83 PTGDR2 (0.49) PTGDR2CYP2C9PTGDR
SCHEMBL21031946 0.80 PTGDR2 (0.53) PTGDR2CYP2C9PTGDR
SCHEMBL21032557 0.80 PTGDR2 (0.54) PTGDR2CYP2C9PTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489233-B1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD (CN) 2022-01-12 EP disclosed
EP-3489233-A1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2019-05-29 EP disclosed