SCHEMBL21032161

SCHEMBL21032161

COC(OC)c1c(C#N)cc(Cl)nc1Nc1cccc(C)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
NFKB1 P19838 1/20 0.41
EGFR P00533 2/20 0.40
ERBB2 P04626 1/20 0.40
KDM4E B2RXH2 4/20 0.40
MAPT P10636 2/20 0.40
GAA P10253 1/20 0.40
FER P16591 5/20 0.40
RXFP1 Q9HBX9 2/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.39
IMPDH2 P12268 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1986224 0.79 FER (0.46) KMT2ANFKB1EGFRERBB2MAPT
SCHEMBL22475481 0.77 FER (0.43) KMT2ANFKB1EGFRMAPTGAA
SCHEMBL30041532 0.71 EGFR (0.57) KMT2ANFKB1EGFRERBB2KDM4E
SCHEMBL26101728 0.71 EGFR (0.57) KMT2ANFKB1EGFRERBB2KDM4E
SCHEMBL28257227 0.69 KMT2A (0.53) KMT2ANFKB1EGFRKDM4EMAPT
SCHEMBL12755667 0.67 NFKB1 (0.55) KMT2ANFKB1EGFRKDM4EMAPT
SCHEMBL30041610 0.65 EGFR (0.50) KMT2AEGFRERBB2KDM4ELMNA
SCHEMBL1986212 0.65 EGFR (0.44) KMT2AEGFRERBB2MAPTMEN1
SCHEMBL19790518 0.65 AURKA (0.49) KMT2AKDM4EMAPTGAAFER
SCHEMBL10254010 0.65 NFKB1 (0.49) NFKB1MAPTFERLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489236-A1 PROCESS FOR THE PREPARATION OF FUSED HETEROAROMATIC PYRROLIDINONES Takeda Pharmaceutical Company Limited (JP) 2019-05-29 EP disclosed