SCHEMBL21032471

SCHEMBL21032471

Cc1c(-c2csc3ccc(Cl)cc23)c2cc(Cl)ccc2n1CC(=O)O

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 19/20 0.57
PTGS1 P23219 1/20 0.56
AKR1B1 P15121 3/20 0.49
CYP2C9 P11712 1/20 0.48
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21031945 0.96 PTGDR2 (0.63) PTGDR2PTGS1AKR1B1CYP2C9
SCHEMBL24180036 0.96 PTGDR2 (0.63) PTGDR2PTGS1AKR1B1CYP2C9
SCHEMBL21032166 0.95 PTGDR2 (0.59) PTGDR2PTGS1AKR1B1CYP2C9
SCHEMBL317472 0.92 PTGDR2 (0.57) PTGDR2PTGS1AKR1B1CYP2C9
SCHEMBL21032558 0.92 PTGDR2 (0.56) PTGDR2PTGS1AKR1B1KEAP1NFE2L2
SCHEMBL21031879 0.90 PTGDR2 (0.52) PTGDR2PTGS1AKR1B1
SCHEMBL21032884 0.87 PTGDR2 (0.53) PTGDR2PTGS1AKR1B1CYP2C9
SCHEMBL24179951 0.87 PTGDR2 (0.56) PTGDR2AKR1B1CYP2C9
SCHEMBL21032561 0.86 PTGDR2 (0.59) PTGDR2PTGS1AKR1B1CYP2C9
SCHEMBL21032209 0.85 PTGDR2 (0.61) PTGDR2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489233-B1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD (CN) 2022-01-12 EP disclosed
EP-3489233-A1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2019-05-29 EP disclosed