SCHEMBL21034692

SCHEMBL21034692

Clc1ccc2[nH]c(CC3CCCCC3)nc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.54
AAK1 Q2M2I8 1/20 0.51
CACNA1H O95180 3/20 0.48
CACNA1G O43497 2/20 0.48
PDE9A O76083 1/20 0.46
TDP1 Q9NUW8 1/20 0.44
RIPK1 Q13546 1/20 0.44
CCNB2 O95067 1/20 0.42
CDK1 P06493 1/20 0.42
CCNB1 P14635 1/20 0.42
GSK3A P49840 1/20 0.42
GSK3B P49841 1/20 0.42
CCNB3 Q8WWL7 1/20 0.42
HRH4 Q9H3N8 1/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
OPRL1 P41146 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8809271 0.82 AAK1 (0.51) IDO1AAK1CACNA1HCACNA1GTDP1
SCHEMBL17516021 0.82 AAK1 (0.51) IDO1AAK1CACNA1HCACNA1GLMNA
SCHEMBL21034524 0.82 AAK1 (0.51) IDO1AAK1CACNA1HCACNA1GLMNA
SCHEMBL21034198 0.81 IDO1 (0.82) IDO1CACNA1HCACNA1G
SCHEMBL21034384 0.81 IDO1 (0.82) IDO1CACNA1HCACNA1G
SCHEMBL21034383 0.81 IDO1 (0.82) IDO1CACNA1HCACNA1G
SCHEMBL21034172 0.81 IDO1 (0.57) IDO1AAK1CACNA1HCACNA1GLMNA
SCHEMBL21034102 0.80 IDO1 (0.65) IDO1AAK1CACNA1HCACNA1GTDP1
SCHEMBL21035054 0.79 AAK1 (0.48) IDO1AAK1CACNA1HCACNA1GCCNB2
SCHEMBL21035092 0.79 IDO1 (0.57) IDO1AAK1CACNA1HCACNA1GLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019101188-A1 NOVEL BENZOIMIDAZOLES AS SELECTIVE INHIBITORS OF INDOLEAMINE 2, 3-DIOXYGENASES BEIGENE, LTD. (GB) 2019-05-31 WO disclosed