SCHEMBL21035528

SCHEMBL21035528

ClCc1ccc(-c2ccc(Cl)cn2)nc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
GRM5 P41594 1/20 0.36
GRM2 Q14416 1/20 0.36
CNR2 P34972 1/20 0.36
HDAC1 Q13547 1/20 0.35
RAB9A P51151 1/20 0.34
CASP3 P42574 1/20 0.34
CCR1 P32246 1/20 0.33
CCR5 P51681 1/20 0.33
CCR8 P51685 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28288104 0.89 CCR1 (0.40) RAB9ACCR1CCR5CCR8HDAC6
SCHEMBL30888429 0.89 CCR1 (0.40) RAB9ACCR1CCR5CCR8HDAC6
SCHEMBL1549465 0.84 GRM2 (0.50) KDM4EGRM2RAB9ACASP3
SCHEMBL21035108 0.84 CNR2 (0.44) KDM4EGRM2CNR2RAB9A
SCHEMBL197456 0.82 CCR1 (0.46) GRM5CNR2CASP3CCR1CCR5
SCHEMBL31504098 0.82 CCR1 (0.46) GRM5CNR2CASP3CCR1CCR5
Hydrochloric Acid SCHEMBL7040410 0.75 KDM4E (0.52) KDM4ERAB9ACCR1CCR5CCR8
SCHEMBL2411349 0.73 CYP11B1 (0.59) RAB9A
SCHEMBL17799 0.73
SCHEMBL21873406 0.72 KMT2A (0.39) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019104011-A1 CERAMIDE GALACTOSYLTRANSFERASE INHIBITORS FOR THE TREATMENT OF DISEASE BIOMARIN PHARMACEUTICAL INC. (US) 2019-05-31 WO disclosed