SCHEMBL21035638

SCHEMBL21035638

NC1CCN(C(=O)[C@@H]2CN(Cc3ccc(-c4ccc(OC(F)(F)F)cc4)nc3)CCN2S(=O)(=O)c2ccc(OCC3CCCCC3)cc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 9/20 0.40
TRPA1 O75762 3/20 0.39
MMP1 P03956 2/20 0.38
MMP9 P14780 2/20 0.38
MMP13 P45452 2/20 0.38
ADAM17 P78536 1/20 0.38
PRKAA2 P54646 1/20 0.37
STAT3 P40763 2/20 0.37
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21034961 0.97 GHSR (0.40) GHSRTRPA1MMP1MMP9MMP13
Trifluoroacetic Acid SCHEMBL21002076 0.94 GHSR (0.40) GHSRTRPA1MMP1MMP9MMP13
Trifluoroacetic Acid SCHEMBL21002077 0.94 GHSR (0.40) GHSRTRPA1MMP1MMP9MMP13
SCHEMBL21035509 0.93 KCNQ1 (0.40) GHSRMMP1MMP9MMP13ADAM17
SCHEMBL21035506 0.93 GHSR (0.44) GHSRMMP1MMP9MMP13ADAM17
SCHEMBL21002178 0.93 GHSR (0.44) GHSRMMP1MMP9MMP13ADAM17
SCHEMBL21002181 0.93 GHSR (0.44) GHSRMMP1MMP9MMP13ADAM17
SCHEMBL21036230 0.91 GHSR (0.44) GHSRMMP1MMP9MMP13ADAM17
Trifluoroacetic Acid SCHEMBL21001843 0.91 GHSR (0.40) GHSRMMP1MMP9MMP13ADAM17
SCHEMBL21034974 0.90 GHSR (0.44) GHSRMMP1MMP9MMP13ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019104011-A1 CERAMIDE GALACTOSYLTRANSFERASE INHIBITORS FOR THE TREATMENT OF DISEASE BIOMARIN PHARMACEUTICAL INC. (US) 2019-05-31 WO disclosed