Etaconazole

Etaconazole

SCHEMBL21043

CCC1COC(Cn2cncn2)(c2ccc(Cl)cc2Cl)O1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 16/20 1.00
THRB P10828 1/20 1.00
LMNA P02545 2/20 0.63
FYN P06241 2/20 0.63
CYP51A1 Q16850 2/20 0.63
HSP90AA1 P07900 2/20 0.63
ADRA1A P35348 2/20 0.63
NR1I2 O75469 1/20 0.63
PGR P06401 1/20 0.63
CHRM2 P08172 1/20 0.63
CHRM4 P08173 1/20 0.63
CHRM5 P08912 1/20 0.63
ADRA2A P08913 1/20 0.63
CHRM1 P11229 1/20 0.63
TSHR P16473 1/20 0.63
ADRA2B P18089 1/20 0.63
ADRA2C P18825 1/20 0.63
CHRM3 P20309 1/20 0.63
DRD1 P21728 1/20 0.63
TBXA2R P21731 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Etaconazole SCHEMBL14884463 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL14884464 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL29827140 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL29386134 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL14884461 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL23421942 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL14884462 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Propiconazole SCHEMBL2522027 0.93 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Propiconazole SCHEMBL5598958 0.93 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Propiconazole SCHEMBL30149161 0.93 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 13239 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026105160-A1 NOVEL AGROCHEMICAL COMPOSITION COMPRISING 3-SUBSTITUTED PHENYLAMIDINE COMPOUNDS AND USE THEREOF PI INDUSTRIES LTD. (IN) 2026-05-21 WO claimed
US-20260101900-A1 OIL LIQUID FUNGICIDAL FORMULATION ADAMA MAKHTESHIM LTD. (IL) 2026-04-16 US claimed
US-20260076371-A1 AGROCHEMICAL COMPOSITION OF TRIAZOLES ADAMA MAKHTESHIM LTD. (IL) 2026-03-19 US claimed
WO-2026041871-A1 METHODS OF CONTROLLING CAUSAL AGENTS OF RAMULARIA LEAF SPOT OR RHYNCHOSPORIUM LEAF SCALD DISEASE, AND COMPOSITIONS FOR THE SAME GOWAN CROP PROTECTION LIMITED (GB) 2026-02-26 WO claimed
EP-4114183-B1 FUNGICIDAL COMPOSITIONS SYNGENTA CROP PROTECTION AG (CH) 2026-02-25 EP claimed
US-20260026501-A1 AGROCHEMICAL COMPOSITION OF SDHI FUNGICIDES ADAMA MAKHTESHIM LTD. (IL) 2026-01-29 US claimed
EP-4654820-A1 FUNGICIDAL COMBINATION UPL Mauritius Limited (MU) 2025-12-03 EP claimed
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
US-20250351828-A1 AZOLE FUNGICIDE COMPOSITION ADAMA MAKHTESHIM LTD. (IL) 2025-11-20 US claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
EP-0209234-A2 Synergistic fungicidal composition UNIROYAL LIMITED (GB) 1987-01-21 EP claimed
EP-0180263-A3 METHOD FOR CONTROLLING VASCULAR WITHERING DISEASES IN PLANTS, ESPECIALLY DUTCH ELM DISEASE Nederlandse Organisatie voor toegepast-natuurwetenschappelijk onderzoek TNO (NL) 1986-07-30 EP claimed
EP-0180263-A2 Method for controlling vascular withering diseases in plants, especially dutch elm disease Nederlandse Organisatie voor toegepast-natuurwetenschappelijk onderzoek TNO (NL) 1986-05-07 EP claimed
US-4542146-A Process for the protection of wood and coatings against deterioration by microorganisms JANSSEN PHARMACEUTICA N.V. (BE) 1985-09-17 US claimed
EP-0038109-B1 AGENTS AND METHOD FOR THE PROTECTION OF COATINGS AND WOOD AND OTHER NON-LIVING ORGANIC SUBSTRATES FROM DETERIORATION BY MICRO-ORGANISMS JANSSEN PHARMACEUTICA N.V. (BE) 1984-08-29 EP claimed
EP-0101102-A2 Preventing fungal decay of food products, particularly harvested fruits JANSSEN PHARMACEUTICA N.V. (BE) 1984-02-22 EP claimed
US-4391813-A 1-//2-/2,4-DICHLOROPHENYL/-4-ETHYL-1,3-DIOXOLAN-2-YL/METHYL/-1H-1,2,4-TRIAZOLE CORNELL RESEARCH FOUNDATION, INC. (US) 1983-07-05 US claimed
EP-0038109-A2 Agents and method for the protection of coatings and wood and other non-living organic substrates from deterioration by micro-organisms JANSSEN PHARMACEUTICA N.V. (BE) 1981-10-21 EP claimed
US-4160838-A FUNGICIDES, BACTERICIDES JANSSEN PHARMACEUTICA N.V. (BE) 1979-07-10 US claimed
US-4079062-A ANTIMICROBIAL, PLANT GROWTH REGULATORS; 1-(B-ARYL)ETHYL-1H-1,2,4-TRIAZOLE KETALS JANSSEN PHARMACEUTICA N.V. (BE) 1978-03-14 US claimed