Etaconazole

Etaconazole

SCHEMBL29827140

CCC1CO[C@](Cn2cncn2)(c2ccc(Cl)cc2Cl)O1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 16/20 1.00
THRB P10828 1/20 1.00
LMNA P02545 2/20 0.63
FYN P06241 2/20 0.63
CYP51A1 Q16850 2/20 0.63
HSP90AA1 P07900 2/20 0.63
ADRA1A P35348 2/20 0.63
NR1I2 O75469 1/20 0.63
PGR P06401 1/20 0.63
CHRM2 P08172 1/20 0.63
CHRM4 P08173 1/20 0.63
CHRM5 P08912 1/20 0.63
ADRA2A P08913 1/20 0.63
CHRM1 P11229 1/20 0.63
TSHR P16473 1/20 0.63
ADRA2B P18089 1/20 0.63
ADRA2C P18825 1/20 0.63
CHRM3 P20309 1/20 0.63
DRD1 P21728 1/20 0.63
TBXA2R P21731 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Etaconazole SCHEMBL14884463 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL21043 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL14884464 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL29386134 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL14884461 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL23421942 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Etaconazole SCHEMBL14884462 1.00 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Propiconazole SCHEMBL2522027 0.93 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Propiconazole SCHEMBL5598958 0.93 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1
Propiconazole SCHEMBL30149161 0.93 CYP3A4 (1.00) CYP3A4THRBLMNAFYNCYP51A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025090255-A1 EMULSION CONCENTRATES, WOOD PRESERVATIVE COMPOSITIONS FORMED THEREFROM, METHODS OF MANUFACTURE THEREOF, AND METHODS OF USE THEREOF KOPPERS PERFORMANCE CHEMICALS, INC. (US) 2025-05-01 WO disclosed
EP-4380364-A1 A WOOD PRESERVATIVE COMPOSITION COMPRISING 4,5-DICHLORO-2-OCTYLISOTHIAZOL-3(2H)-ONE, A METHOD TREATING A WOOD SUBSTRATE THEREWITH, AND A WOOD PRODUCT PRODUCED THEREFROM Koppers Performance Chemicals, Inc. (US) 2024-06-12 EP disclosed
EP-4380365-A1 A WOOD PRESERVATIVE COMPOSITION COMPRISING 4,5-DICHLORO-2-OCTYLISOTHIAZOL-3(2H)-ONE, A METHOD TREATING A WOOD SUBSTRATE THEREWITH, AND A WOOD PRODUCT PRODUCED THEREFROM Koppers Performance Chemicals Inc. (US) 2024-06-12 EP disclosed
EP-4284773-A1 A METHOD FOR PRODUCING COPPER CARBOXYLATE, A WOOD PRESERVATIVE COMPOSITION COMPRISING COPPER CARBOXYLATE, AND A WOOD PRODUCT PRODUCED THEREFROM Koppers Performance Chemicals Inc. (US) 2023-12-06 EP disclosed
WO-2023015302-A1 A WOOD PRESERVATIVE COMPOSITION COMPRISING 4,5-DICHLORO-2-OCTYLISOTHIAZOL-3(2H)-ONE, A METHOD TREATING A WOOD SUBSTRATE THEREWITH, AND A WOOD PRODUCT PRODUCED THEREFROM KOPPERS PERFORMANCE CHEMICALS, INC. (US) 2023-02-09 WO disclosed
WO-2023015305-A1 A WOOD PRESERVATIVE COMPOSITION COMPRISING 4,5-DICHLORO-2-OCTYLISOTHIAZOL-3(2H)-ONE, A METHOD TREATING A WOOD SUBSTRATE THEREWITH, AND A WOOD PRODUCT PRODUCED THEREFROM KOPPERS PERFORMANCE CHEMICALS, INC. (US) 2023-02-09 WO disclosed
WO-2022164532-A1 A METHOD FOR PRODUCING COPPER CARBOXYLATE, A WOOD PRESERVATIVE COMPOSITION COMPRISING COPPER CARBOXYLATE, AND A WOOD PRODUCT PRODUCED THEREFROM KOPPERS PERFORMANCE CHEMICALS, INC. (US) 2022-08-04 WO disclosed