SCHEMBL21043237

SCHEMBL21043237

NC(O)CC1CCCN1C(=O)c1ccc(-c2ccc(OCC3CCN(CC(F)(F)C(F)(F)F)CC3)cn2)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 6/20 0.35
ALOX5AP P20292 2/20 0.35
FEN1 P39748 2/20 0.35
MET P08581 3/20 0.34
POLB P06746 1/20 0.34
CYP4F2 P78329 4/20 0.34
CYP4A11 Q02928 4/20 0.34
PDK2 Q15119 1/20 0.34
HCRTR1 O43613 1/20 0.33
ROCK2 O75116 1/20 0.33
PDE4B Q07343 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18848900 0.88 PDK2 (0.41) GPR119CYP4F2CYP4A11PDK2
SCHEMBL16758018 0.87 PDK2 (0.42) GPR119CYP4F2CYP4A11PDK2
SCHEMBL16758023 0.87 PDK2 (0.42) GPR119CYP4F2CYP4A11PDK2
SCHEMBL18849010 0.84 GPR119 (0.43) GPR119CYP4F2CYP4A11
SCHEMBL15539479 0.83 POLB (0.46) GPR119ALOX5APFEN1POLBCYP4F2
SCHEMBL15539188 0.83 POLB (0.46) GPR119ALOX5APFEN1POLBCYP4F2
SCHEMBL15539187 0.83 POLB (0.46) GPR119ALOX5APFEN1POLBCYP4F2
SCHEMBL16757844 0.82 CYP4F2 (0.41) GPR119CYP4F2CYP4A11
SCHEMBL16758060 0.81 CNR2 (0.39) GPR119CYP4F2CYP4A11PDK2
SCHEMBL16758055 0.81 CNR2 (0.39) GPR119CYP4F2CYP4A11PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3074384-B1 AMIDE DERIVATIVES FOR GPR119 AGONIST CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2019-05-22 EP disclosed