SCHEMBL21044728

SCHEMBL21044728

O=C(NCc1ccc(F)cc1)c1ccc2ccccc2c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 2/20 0.76
HDAC3 O15379 2/20 0.74
HDAC1 Q13547 2/20 0.74
HDAC2 Q92769 2/20 0.74
HDAC4 P56524 1/20 0.74
HDAC7 Q8WUI4 1/20 0.74
HDAC10 Q969S8 1/20 0.74
HDAC11 Q96DB2 1/20 0.74
HDAC8 Q9BY41 1/20 0.74
HDAC6 Q9UBN7 1/20 0.74
HDAC9 Q9UKV0 1/20 0.74
HDAC5 Q9UQL6 1/20 0.74
PPARG P37231 1/20 0.57
NPC1 O15118 1/20 0.57
TP53 P04637 1/20 0.57
MAPT P10636 1/20 0.57
HPGD P15428 1/20 0.57
TSHR P16473 1/20 0.57
RAB9A P51151 1/20 0.57
CXCR4 P61073 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3030027 0.88 HDAC6 (0.74) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL14894197 0.88 NR1H4 (0.85) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL3024525 0.87 HDAC6 (0.72) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL7322242 0.87 NR1H4 (1.00) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL4153362 0.86 NPC1 (0.69) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL8243848 0.85 NR1H4 (0.76) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL14885209 0.85 NR1H4 (0.76) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL28918342 0.85 HDAC1 (0.79) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL10207296 0.85 HDAC6 (1.00) NR1H4HDAC3HDAC1HDAC2HDAC4
SCHEMBL3031645 0.85 MAPT (0.58) NR1H4HDAC3HDAC1HDAC2HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3284520-B1 POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING HIV INTEGRASE INHIBITORY ACTIVITY VIIV HEALTHCARE CO (US) 2019-06-05 EP disclosed