SCHEMBL28918342

SCHEMBL28918342

NNC(=O)c1ccc(CNC(=O)c2ccc3ccccc3c2)cc1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.79
HDAC6 Q9UBN7 5/20 0.79
HDAC2 Q92769 4/20 0.79
HDAC3 O15379 3/20 0.79
HDAC8 Q9BY41 3/20 0.79
HDAC4 P56524 2/20 0.79
HDAC7 Q8WUI4 2/20 0.79
HDAC10 Q969S8 2/20 0.79
HDAC11 Q96DB2 2/20 0.79
HDAC9 Q9UKV0 2/20 0.79
HDAC5 Q9UQL6 2/20 0.79
NR1H4 Q96RI1 4/20 0.76
NPC1 O15118 2/20 0.60
MAPT P10636 2/20 0.60
HPGD P15428 2/20 0.57
TP53 P04637 1/20 0.57
TSHR P16473 1/20 0.57
RAB9A P51151 1/20 0.57
PLAU P00749 1/20 0.54
EPHX2 P34913 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10207296 0.88 HDAC6 (1.00) HDAC1HDAC6HDAC2HDAC3HDAC8
SCHEMBL14885209 0.88 NR1H4 (0.76) HDAC1HDAC6HDAC2HDAC3HDAC8
SCHEMBL14894197 0.88 NR1H4 (0.85) HDAC1HDAC6HDAC2HDAC3HDAC8
SCHEMBL12588095 0.87 HDAC1 (0.77) HDAC1HDAC6HDAC2HDAC3HDAC8
SCHEMBL7322242 0.87 NR1H4 (1.00) HDAC1HDAC6HDAC2HDAC3HDAC8
SCHEMBL1149678 0.86 NPC1 (0.62) HDAC1HDAC6HDAC2HDAC3HDAC8
SCHEMBL8243848 0.85 NR1H4 (0.76) HDAC1HDAC6HDAC2HDAC3HDAC8
SCHEMBL21044728 0.85 NR1H4 (0.76) HDAC1HDAC6HDAC2HDAC3HDAC8
SCHEMBL21454774 0.84 HDAC6 (0.75) HDAC1HDAC6HDAC2HDAC3HDAC8
SCHEMBL11902028 0.84 NR1H4 (0.79) HDAC1HDAC6HDAC2HDAC3HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113831338-B Histone deacetylase inhibitor and preparation method and application thereof 中国海洋大学 2022-12-20 CN disclosed