SCHEMBL21048435

SCHEMBL21048435

[O-][S+](C=CCCN=C=S)c1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
XPO1 O14980 1/20 0.40
KEAP1 Q14145 2/20 0.38
NFE2L2 Q16236 2/20 0.38
TRPA1 O75762 2/20 0.33
CYP2E1 P05181 1/20 0.33
CYP2A6 P11509 1/20 0.33
MIF P14174 1/20 0.33
HIF1A Q16665 1/20 0.33
CYP2A13 Q16696 1/20 0.33
EPAS1 Q99814 1/20 0.33
NAAA Q02083 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19822506 1.00 XPO1 (0.40) XPO1KEAP1NFE2L2TRPA1CYP2E1
SCHEMBL21048436 0.83 XPO1 (0.52) XPO1KEAP1NFE2L2TRPA1CYP2E1
SCHEMBL19822504 0.83 XPO1 (0.52) XPO1KEAP1NFE2L2TRPA1CYP2E1
SCHEMBL19822514 0.78 XPO1 (0.34) XPO1
SCHEMBL21048406 0.76 NAAA (0.36) XPO1HIF1ANAAA
SCHEMBL21048405 0.76 XPO1 (0.48) XPO1KEAP1NFE2L2TRPA1CYP2E1
SCHEMBL19822524 0.76 XPO1 (0.48) XPO1KEAP1NFE2L2TRPA1CYP2E1
SCHEMBL21048404 0.75 XPO1 (0.40) XPO1TRPA1CYP2E1CYP2A6MIF
SCHEMBL19822516 0.75 XPO1 (0.40) XPO1TRPA1CYP2E1CYP2A6MIF
SCHEMBL21048407 0.75 XPO1 (0.44) XPO1MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10315990-B2 Isothiocyanate compounds and isothiocyanate XPO1 protein inhibitor drugs thereof DRIVINGFORCE THERAPEUTICS (CN) 2019-06-11 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10315990-B2 Isothiocyanate compounds and isothiocyanate XPO1 protein inhibitor drugs thereof XPO1, XPOT, XPO4 XPO1 1/4885KEAP1 10/4885NFE2L2 75/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.