SCHEMBL21056103

SCHEMBL21056103

C/C(C#N)=C\c1cc(C)cc(C)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.49
GABRG2 P18507 2/20 0.49
GABRB3 P28472 2/20 0.49
EGFR P00533 8/20 0.39
ERBB2 P04626 4/20 0.39
MAPT P10636 5/20 0.38
CYP2C9 P11712 4/20 0.38
CYP2C19 P33261 2/20 0.38
HPGD P15428 4/20 0.37
ALDH1A1 P00352 5/20 0.36
KMT2A Q03164 5/20 0.36
MEN1 O00255 4/20 0.36
LMNA P02545 4/20 0.36
RGS12 O14924 3/20 0.36
CYP3A4 P08684 3/20 0.36
ALOX15 P16050 3/20 0.36
NFKB1 P19838 3/20 0.36
BLM P54132 3/20 0.36
GNAI1 P63096 3/20 0.36
PMP22 Q01453 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21134491 1.00 GABRA1 (0.49) GABRA1GABRG2GABRB3EGFRERBB2
SCHEMBL21056104 1.00 GABRA1 (0.49) GABRA1GABRG2GABRB3EGFRERBB2
SCHEMBL26552257 0.82 RPS6KA3 (0.48) GABRA1GABRG2GABRB3EGFRERBB2
SCHEMBL13681565 0.81 EGFR (0.46) GABRA1GABRG2GABRB3EGFRERBB2
SCHEMBL26552237 0.80 GABRA1 (0.51) GABRA1GABRG2GABRB3MAPTALDH1A1
SCHEMBL12755365 0.78 GABRA1 (0.53) GABRA1GABRG2GABRB3EGFRERBB2
SCHEMBL11957026 0.78 GABRA1 (0.53) GABRA1GABRG2GABRB3EGFRERBB2
SCHEMBL13908793 0.78 GABRA1 (0.53) GABRA1GABRG2GABRB3EGFRERBB2
SCHEMBL12715623 0.78 GABRA1 (0.45) GABRA1GABRG2GABRB3EGFRERBB2
SCHEMBL17884073 0.78 EGFR (0.43) GABRA1GABRG2GABRB3EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3498273-A1 PHARMACEUTICAL COMPOSITION FOR MODULATING THE RESPONSE OF A GABA-A RECEPTOR Universität Wien (AT) 2019-06-19 EP disclosed
EP-3498273-A1 PHARMACEUTICAL COMPOSITION FOR MODULATING THE RESPONSE OF A GABA-A RECEPTOR Universität Wien (AT) 2019-06-19 EP disclosed