SCHEMBL2106264

SCHEMBL2106264

c1cc(C2=Nc3ccccc3CO2)cc(C2CC2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.40
CYP2D6 P10635 1/20 0.35
MEN1 O00255 1/20 0.35
RECQL P46063 1/20 0.35
KMT2A Q03164 1/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
KCNH2 Q12809 1/20 0.34
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
HTR2C P28335 4/20 0.32
BACE1 P56817 1/20 0.31
GRIN2B Q13224 2/20 0.31
NR3C1 P04150 1/20 0.31
PGR P06401 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18100313 0.85 NPC1 (0.42) KMT2ANPC1RAB9AKDM4EALDH1A1
SCHEMBL10654837 0.78 NPC1 (0.49) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL28137726 0.78 NPC1 (0.41) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL28574627 0.78 NPC1 (0.41) NOTUMMEN1KMT2ANPC1RAB9A
SCHEMBL11907198 0.77 NPC1 (0.42) CYP2D6MEN1RECQLKMT2ANPC1
SCHEMBL30129926 0.77 NPC1 (0.42) CYP2D6MEN1RECQLKMT2ANPC1
SCHEMBL28138209 0.75 KDM4E (0.38) NPC1RAB9AKDM4EALDH1A1LMNA
SCHEMBL28579741 0.72 MAPT (0.36) NOTUMNPC1RAB9AKDM4EALDH1A1
SCHEMBL28569090 0.70 MAPT (0.43) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL28915334 0.70 NPC1 (0.42) KMT2ANPC1RAB9AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163740-B2 6-substituted benzoxazines HOFFMANN-LA ROCHE INC. (US) 2012-04-24 US disclosed