SCHEMBL21075937

SCHEMBL21075937

CC(F)(F)c1ccc(Cc2c(N3CCC3)nc3ccc(Br)cc3c2F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 8/20 0.41
ALDH1A1 P00352 4/20 0.36
KDM4E B2RXH2 2/20 0.36
LMNA P02545 2/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP1A2 P05177 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MITF O75030 1/20 0.35
ALPG P10696 1/20 0.35
HTT P42858 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CYP3A4 P08684 1/20 0.33
PTGFR P43088 1/20 0.33
CTNNB1 P35222 1/20 0.33
TCF7L2 Q9NQB0 1/20 0.33
NPY5R Q15761 1/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16632658 0.80 RORC (0.57) RORCCYP1A2CTNNB1TCF7L2
SCHEMBL16632413 0.67 RORC (0.55) RORC
SCHEMBL16460911 0.64 CYP1A2 (0.45) RORCALDH1A1KDM4ELMNAMAPT
SCHEMBL16462100 0.64 CYP1A2 (0.61) RORCCYP1A2
SCHEMBL15647927 0.63 RORC (0.47) RORCCYP1A2
SCHEMBL21574565 0.63 CYP1A2 (0.41) RORCALDH1A1KDM4ELMNAKMT2A
SCHEMBL16460893 0.62 RORC (0.41) RORCALDH1A1KDM4ELMNAMAPT
SCHEMBL15648267 0.62 CYP1A2 (0.52) RORCCYP1A2
Hydrochloric Acid SCHEMBL5578269 0.62 KDM4E (0.74) ALDH1A1KDM4ELMNAMAPTKMT2A
SCHEMBL15647695 0.62 RORC (0.63) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057949-B1 SECONDARY ALCOHOL QUINOLINYL MODULATORS OF ROR GAMMA T JANSSEN PHARMACEUTICA NV (BE) 2019-06-05 EP disclosed