SCHEMBL21077210

SCHEMBL21077210

CCC(C(=O)N(C)c1ccc(-c2cncc(C#N)c2)cc1)c1csc(NSC2CC2)n1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTPS1 P17812 5/20 0.42
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36
PIK3CG P48736 1/20 0.36
GPR119 Q8TDV5 1/20 0.35
XDH P47989 1/20 0.34
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
GRIA2 P42262 1/20 0.33
KDM4E B2RXH2 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
CHRM1 P11229 1/20 0.32
BRD4 O60885 1/20 0.30
CREBBP Q92793 1/20 0.30
KDM1A O60341 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21044272 0.86 CTPS1 (0.55) CTPS1
SCHEMBL21077181 0.85 CTPS1 (0.39) CTPS1KDM4E
SCHEMBL21077201 0.82 CTPS1 (0.48) CTPS1GSK3BDYRK1APIK3CG
SCHEMBL21076874 0.73 CTPS1 (0.45) CTPS1GSK3BDYRK1APIK3CG
SCHEMBL21044260 0.72 CTPS1 (0.73) CTPS1
SCHEMBL21077225 0.71 CTPS1 (0.43) CTPS1KDM4E
SCHEMBL21077144 0.71 CTPS1 (0.55) CTPS1GSK3BDYRK1APIK3CGXDH
SCHEMBL21044425 0.70 CTPS1 (0.56) CTPS1
SCHEMBL22762461 0.69 CTPS1 (0.55) CTPS1KDM4E
SCHEMBL30529007 0.68 CTPS1 (0.59) CTPS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3492454-A1 COMPOUNDS Step Pharma S.A.S. (FR) 2019-06-05 EP disclosed