SCHEMBL21077907

SCHEMBL21077907

N#CCCC1(c2ccc(O)cc2)CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.47
ESR2 Q92731 2/20 0.47
TSHR P16473 1/20 0.43
HTT P42858 1/20 0.43
EPHX2 P34913 1/20 0.39
HSD17B10 Q99714 1/20 0.38
SLC6A3 Q01959 9/20 0.38
SLC6A4 P31645 7/20 0.38
HSD11B1 P28845 1/20 0.37
SLC6A2 P23975 4/20 0.36
CYP19A1 P11511 1/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28309415 0.80 ESR1 (0.55) ESR1ESR2SLC6A3SLC6A4HSD11B1
SCHEMBL18440458 0.77 TSHR (0.58) TSHRHTTEPHX2HSD17B10SLC6A3
SCHEMBL12002346 0.77 ESR1 (0.52) ESR1ESR2SLC6A3SLC6A4HSD11B1
SCHEMBL8735345 0.76 ESR1 (0.59) ESR1ESR2SLC6A3SLC6A4HSD11B1
SCHEMBL5682331 0.75 CNR2 (0.52) ESR1ESR2SLC6A3SLC6A4SLC6A2
SCHEMBL8706024 0.74 ESR2 (0.57) ESR1ESR2SLC6A3SLC6A4HSD11B1
SCHEMBL12000487 0.73 ESR1 (0.47) ESR1ESR2SLC6A3SLC6A4HSD11B1
SCHEMBL4564526 0.73 CNR2 (0.58) ESR1ESR2HSD17B10SLC6A3SLC6A4
SCHEMBL10791207 0.73 ESR1 (0.55) ESR1ESR2SLC6A3SLC6A4SLC6A2
SCHEMBL5678460 0.72 CNR2 (0.60) ESR1ESR2HSD17B10SLC6A3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041841-B1 TRIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND METHODS OF USE THEREOF HOFFMANN LA ROCHE (CH) 2019-06-05 EP disclosed