SCHEMBL2108656

SCHEMBL2108656

O=c1c(Cl)c(Cl)sn1Cc1ccc(Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 6/20 0.53
EP300 Q09472 2/20 0.51
CREBBP Q92793 2/20 0.51
KAT2A Q92830 2/20 0.51
MAPT P10636 3/20 0.42
THRB P10828 1/20 0.42
CASP3 P42574 4/20 0.41
FAAH O00519 1/20 0.41
MGLL Q99685 1/20 0.41
VEGFA P15692 1/20 0.40
EGLN1 Q9GZT9 1/20 0.40
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KMT2A Q03164 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
MC4R P32245 1/20 0.39
OPRK1 P41145 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GPR35 Q9HC97 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5593645 0.86 KAT2B (0.50) KAT2BEP300CREBBPKAT2AMAPT
SCHEMBL1876020 0.85 CASP3 (0.57) KAT2BMAPTCASP3FAAHMGLL
SCHEMBL2109324 0.82 MAPT (0.56) KAT2BEP300CREBBPKAT2AMAPT
SCHEMBL8727611 0.82 KAT2B (0.49) KAT2BEP300CREBBPKAT2AMAPT
SCHEMBL14640378 0.80 KAT2B (0.49) KAT2BEP300CREBBPKAT2ACASP3
SCHEMBL5593690 0.80 KAT2B (0.49) KAT2BEP300CREBBPKAT2ACASP3
SCHEMBL5593816 0.79 GAA (0.46) KAT2BEP300CREBBPKAT2ACASP3
SCHEMBL5593705 0.78 HDAC3 (0.46) KAT2BCASP3FAAHMGLLMEN1
SCHEMBL5593642 0.77 MAOB (0.39) KAT2BEP300CREBBPKAT2ARGS4
SCHEMBL5593627 0.76 KMT2A (0.43) KAT2BMAPTFAAHMGLLMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5912286-A Silicone-containing fluoropolymers for controlled release of organic leachants THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1999-06-15 US claimed
EP-0762955-A4 ANTIFOULING AND FOUL-RELEASE COATINGS US HEALTH (US) 1998-01-07 EP claimed
EP-0762955-A1 ANTIFOULING AND FOUL-RELEASE COATINGS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY OF THE NAVY (US) 1997-03-19 EP claimed
WO-1995032862-A1 ANTIFOULING AND FOUL-RELEASE COATINGS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1995-12-07 WO claimed
US-4127687-A PAINTING WITH ISOTHIAZOLONES ROHM AND HAAS COMPANY (US) 1978-11-28 US claimed
US-8157877-B2 Chemical mechanical polishing aqueous dispersion, chemical mechanical polishing method, and kit for preparing chemical mechanical polishing aqueous dispersion JSR CORPORATION (JP) 2012-04-17 US disclosed
US-20090325323-A1 AQUEOUS DISPERSION FOR CHEMICAL MECHANICAL POLISHING, PRODUCTION METHOD THEREOF, AND CHEMICAL MECHANICAL POLISHING METHOD JSR CORPORATION (JP) 2009-12-31 US disclosed
US-20090165395-A1 CHEMICAL MECHANICAL POLISHING AQUEOUS DISPERSION, CHEMICAL MECHANICAL POLISHING METHOD, AND KIT FOR PREPARING CHEMICAL MECHANICAL POLISHING AQUEOUS DISPERSION JSR CORPORATION (JP) 2009-07-02 US disclosed
EP-1962334-A1 AQUEOUS DISPERSION FOR CHEMICAL MECHANICAL POLISHING, CHEMICAL MECHANICAL POLISHING METHOD, AND KIT FOR PREPARING AQUEOUS DISPERSION FOR CHEMICAL MECHANICAL POLISHING JSR Corporation (JP) 2008-08-27 EP disclosed
US-6786944-B2 FOR USE IN MICRO ISOLATING STEP OR A PLANARIZING STEP OF AN INTER LAYER DIELECTRIC IN PRODUCTION OF SEMICONDUCTOR DEVICES JSR CORPORATION (JP) 2004-09-07 US disclosed
EP-1357161-A2 Aqueous dispersion for chemical mechanical polishing JSR Corporation (JP) 2003-10-29 EP disclosed
US-20030196386-A1 Aqueous dispersion for chemical mechanical polishing JSR CORPORATION (JP) 2003-10-23 US disclosed
EP-1059033-A1 INDUSTRIAL ANTIBACTERIAL/ANTIFUNGAL AGENTS, ALGICIDES AND ANTI-BIOLOGICAL ADHESION AGENTS CONTAINING BENZYLAMINES Nissan Chemical Industries, Ltd. (JP) 2000-12-13 EP disclosed
US-6153648-A Iodopropargylamine compounds, and industrial antimicrobial and antifungal agents, algicides, and antifouling agents containing the same NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2000-11-28 US disclosed
EP-1016649-A1 IODOPROPAGYLAMINE COMPOUNDS, AND INDUSTRIAL ANTIMICROBIAL AND ANTIFUNGAL AGENTS, ALGICIDES, AND ANTIFOULING AGENTS CONTAINING THE SAME Nissan Chemical Industries, Ltd. (JP) 2000-07-05 EP disclosed
US-5912286-A Silicone-containing fluoropolymers for controlled release of organic leachants THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1999-06-15 US disclosed
EP-0762955-A4 ANTIFOULING AND FOUL-RELEASE COATINGS US HEALTH (US) 1998-01-07 EP disclosed
EP-0762955-A1 ANTIFOULING AND FOUL-RELEASE COATINGS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY OF THE NAVY (US) 1997-03-19 EP disclosed
WO-1995032862-A1 ANTIFOULING AND FOUL-RELEASE COATINGS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1995-12-07 WO disclosed