SCHEMBL21096776

SCHEMBL21096776

CCOC(=O)c1cnc2nc(C)[nH]c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.49
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
SIRT2 Q8IXJ6 3/20 0.44
SIRT1 Q96EB6 2/20 0.44
PKN1 Q16512 1/20 0.43
PKN2 Q16513 1/20 0.43
ALDH1A1 P00352 3/20 0.43
MAPT P10636 3/20 0.43
RAB9A P51151 2/20 0.43
PPARG P37231 1/20 0.43
NCOA2 Q15596 1/20 0.43
NCOA1 Q15788 1/20 0.43
SIRT3 Q9NTG7 1/20 0.43
MAOB P27338 3/20 0.42
HCRTR1 O43613 2/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21604724 0.80 SMN1; SMN2 (0.56) SMN1; SMN2ALDH1A1RAB9AHPGD
SCHEMBL7214669 0.80 SMN1; SMN2 (0.56) SMN1; SMN2ALDH1A1RAB9AKDM4EMEN1
SCHEMBL4228892 0.78 CYP2C9 (0.48) SMN1; SMN2CYP2C9CYP2C19ALDH1A1MAPT
SCHEMBL6487097 0.75 CA12 (0.46) SMN1; SMN2CYP2C9CYP2C19SIRT2SIRT1
SCHEMBL6169071 0.75 PKN1 (0.67) SMN1; SMN2SIRT2SIRT1PKN1PKN2
SCHEMBL18222953 0.75 ALDH1A1 (0.50) SMN1; SMN2CYP2C9CYP2C19SIRT2SIRT1
SCHEMBL1578883 0.75 CYP2C9 (0.48) CYP2C9CYP2C19RAB9AMAOBCA12
SCHEMBL29827836 0.75 ALDH1A1 (0.50) SMN1; SMN2CYP2C9CYP2C19SIRT2SIRT1
SCHEMBL8832318 0.74 ALDH1A1 (0.43) SMN1; SMN2ALDH1A1MAPTRAB9AKDM4E
SCHEMBL1578888 0.74 CYP2C9 (0.49) SMN1; SMN2CYP2C9CYP2C19ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019116256-A1 FUSED PYRIDINES WHICH ACT AS INHIBITORS OF H-PGDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-06-20 WO disclosed