SCHEMBL2109746

SCHEMBL2109746

CC(C)(C)OC(=O)NNC(=S)c1ccc(F)nc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.40
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
APLNR P35414 1/20 0.38
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP17A1 P05093 2/20 0.36
NAMPT P43490 1/20 0.36
KCNQ3 O43525 1/20 0.35
KCNQ2 O43526 1/20 0.35
EPHX2 P34913 1/20 0.34
MAPT P10636 1/20 0.34
SYK P43405 1/20 0.34
MAPKAPK2 P49137 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2109912 0.85 HDAC1 (0.45) GAAALDH1A1LMNAPOLBAPLNR
SCHEMBL2108776 0.81 GAA (0.44) GAAALDH1A1LMNAPOLBAPLNR
SCHEMBL2108802 0.78 CHRNA1 (0.47) GAAALDH1A1LMNAPOLBAPLNR
SCHEMBL17680521 0.77 SMN1; SMN2 (0.49) GAAALDH1A1LMNAPOLBAPLNR
SCHEMBL30812042 0.76 CA12 (0.43) GAAKCNQ3KCNQ2EPHX2
SCHEMBL646488 0.76 CA12 (0.43) GAAKCNQ3KCNQ2EPHX2
SCHEMBL18654067 0.76 GAA (0.45) GAAALDH1A1LMNAPOLBAPLNR
SCHEMBL24992894 0.74 EPHX2 (0.52) RAB9AEPHX2MAPT
SCHEMBL23747902 0.73 GAA (0.42) GAALMNAPOLBAPLNRMEN1
SCHEMBL392294 0.73 NAMPT (0.51) CYP17A1NAMPTKCNQ3KCNQ2SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8158662-B2 Compounds and compositions as LXR modulators HAMILTON (BM) 2012-04-17 US disclosed
EP-1713799-A2 COMPOUNDS AND COMPOSITIONS AS LXR MODULATORS IRM, LLC (BM) 2006-10-25 EP disclosed
WO-2005077124-A2 COMPOUNDS AND COMPOSITIONS AS LXR MODULATORS IRM LLC (BM) 2005-08-25 WO disclosed