SCHEMBL2109912

SCHEMBL2109912

Cc1ccc(C(=S)NNC(=O)OC(C)(C)C)cn1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
GAA P10253 4/20 0.40
ALDH1A1 P00352 1/20 0.40
NAMPT P43490 2/20 0.39
KDM4E B2RXH2 2/20 0.39
MAPKAPK2 P49137 1/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
DGAT1 O75907 2/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
APLNR P35414 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24599026 0.86 HDAC1 (0.55) HDAC1HDAC6NAMPTKDM4EKMT2A
SCHEMBL2109746 0.85 GAA (0.40) GAAALDH1A1NAMPTMAPKAPK2KMT2A
SCHEMBL16828785 0.78 HDAC1 (0.57) HDAC1HDAC6ALDH1A1NAMPTKDM4E
SCHEMBL17680521 0.78 SMN1; SMN2 (0.49) GAAALDH1A1KMT2AMEN1NPC1
SCHEMBL2108776 0.77 GAA (0.44) GAAALDH1A1KMT2AMEN1NPC1
SCHEMBL9834746 0.76 HDAC1 (0.51) HDAC1HDAC6GAAKDM4EKMT2A
SCHEMBL22770010 0.75 GAA (0.46) HDAC1HDAC6GAAALDH1A1NAMPT
SCHEMBL22558261 0.75 RAB9A (0.57) HDAC1GAAALDH1A1KMT2AMEN1
SCHEMBL10801436 0.74 L3MBTL1 (0.54) HDAC1HDAC6GAAALDH1A1KMT2A
SCHEMBL2108802 0.73 CHRNA1 (0.47) GAAALDH1A1KMT2AMEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8158662-B2 Compounds and compositions as LXR modulators HAMILTON (BM) 2012-04-17 US disclosed
EP-1713799-A2 COMPOUNDS AND COMPOSITIONS AS LXR MODULATORS IRM, LLC (BM) 2006-10-25 EP disclosed
WO-2005077124-A2 COMPOUNDS AND COMPOSITIONS AS LXR MODULATORS IRM LLC (BM) 2005-08-25 WO disclosed