SCHEMBL21098717

SCHEMBL21098717

COc1cc(N2CCNCC2C)ccc1F

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.46
RAD52 P43351 1/20 0.45
HTR2C P28335 8/20 0.41
HTR2A P28223 7/20 0.41
HTR2B P41595 7/20 0.41
ALK Q9UM73 3/20 0.40
MET P08581 1/20 0.40
BRPF1 P55201 2/20 0.39
BRD4 O60885 1/20 0.39
BRD1 O95696 1/20 0.39
BRPF3 Q9ULD4 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21098716 1.00 KDR (0.46) KDRRAD52HTR2CHTR2AHTR2B
SCHEMBL19709333 1.00 KDR (0.46) KDRRAD52HTR2CHTR2AHTR2B
SCHEMBL19709302 0.85 HTR2C (0.42) RAD52HTR2CHTR2AHTR2BBRPF1
SCHEMBL5630952 0.84 RAD52 (0.49) RAD52HTR2CHTR2AHTR2B
SCHEMBL5632465 0.84 RAD52 (0.49) RAD52HTR2CHTR2AHTR2B
SCHEMBL5630960 0.84 RAD52 (0.49) RAD52HTR2CHTR2AHTR2B
SCHEMBL21461789 0.84 ADAMTS5 (0.45) RAD52HTR2CHTR2AHTR2BALK
SCHEMBL19709537 0.84 ADAMTS5 (0.45) RAD52HTR2CHTR2AHTR2BALK
SCHEMBL1639581 0.84 HTR2C (0.48) RAD52HTR2CHTR2AHTR2BSLC6A2
SCHEMBL1639678 0.84 HTR2C (0.48) RAD52HTR2CHTR2AHTR2BSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3498715-B1 ANTI-HCMV VIRUS COMPOUND MEDSHINE DISCOVERY INC (CN) 2021-06-09 EP disclosed
EP-3498715-A1 ANTI-HCMV VIRUS COMPOUND Medshine Discovery Inc. (CN) 2019-06-19 EP disclosed