SCHEMBL21113032

SCHEMBL21113032

CCOc1cc(Cn2c(=O)[nH]c3cc(C(F)(F)F)ccc32)ccc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 2/20 0.51
GRIN1 Q05586 3/20 0.49
GRIN2B Q13224 3/20 0.49
KDM4E B2RXH2 3/20 0.49
NPSR1 Q6W5P4 3/20 0.49
ALDH1A1 P00352 2/20 0.49
HSD17B10 Q99714 2/20 0.47
RAB9A P51151 1/20 0.47
MAOB P27338 1/20 0.45
USP2 O75604 1/20 0.44
GLA P06280 1/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
TP53 P04637 1/20 0.43
HTT P42858 2/20 0.43
TSHR P16473 2/20 0.42
LMNA P02545 1/20 0.42
MEN1 O00255 1/20 0.42
CYP1A2 P05177 1/20 0.42
HSP90AA1 P07900 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21113764 0.86 GRIN1 (0.52) PDE4BGRIN1GRIN2BKDM4ENPSR1
SCHEMBL21113912 0.85 EPHX2 (0.46) PDE4BNPSR1ALDH1A1HSD17B10RAB9A
SCHEMBL22753865 0.84 PDE4B (0.50) PDE4BGRIN1GRIN2BKDM4ENPSR1
SCHEMBL21112114 0.84 PDE4B (0.49) PDE4BGRIN1GRIN2BKDM4ENPSR1
SCHEMBL21115318 0.84 PDE4B (0.50) PDE4BGRIN1GRIN2BKDM4ENPSR1
SCHEMBL21113756 0.83 PDE4B (0.51) PDE4BGRIN1GRIN2BKDM4EALDH1A1
SCHEMBL21113905 0.83 GRIN1 (0.49) PDE4BGRIN1GRIN2BKDM4EALDH1A1
SCHEMBL21113745 0.83 USP2 (0.56) GRIN1GRIN2BKDM4ENPSR1ALDH1A1
SCHEMBL21114090 0.82 HSD17B10 (0.48) PDE4BGRIN1GRIN2BKDM4ENPSR1
SCHEMBL21114204 0.82 SMN1; SMN2 (0.52) KDM4ENPSR1ALDH1A1HSD17B10RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3502099-B1 CYCLIC COMPOUND ACTING AS PDE4 INHIBITOR MEDSHINE DISCOVERY INC (CN) 2020-12-09 EP disclosed
EP-3502099-A1 CYCLIC COMPOUND ACTING AS PDE4 INHIBITOR Medshine Discovery Inc. (CN) 2019-06-26 EP disclosed