SCHEMBL21113745

SCHEMBL21113745

CCOc1cc(Cn2c(=O)[nH]c3ccccc32)ccc1OC

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.56
GLA P06280 1/20 0.56
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 1/20 0.55
HSD17B10 Q99714 1/20 0.54
HTT P42858 4/20 0.54
LMNA P02545 3/20 0.54
TSHR P16473 3/20 0.50
MEN1 O00255 1/20 0.50
CYP1A2 P05177 1/20 0.50
KMT2A Q03164 1/20 0.50
NPSR1 Q6W5P4 1/20 0.49
GRIN1 Q05586 1/20 0.48
GRIN2B Q13224 1/20 0.48
TP53 P04637 1/20 0.47
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21113764 0.85 GRIN1 (0.52) USP2GLAKDM4EALDH1A1HSD17B10
SCHEMBL22753865 0.85 PDE4B (0.50) USP2GLAKDM4EALDH1A1HSD17B10
SCHEMBL21112114 0.85 PDE4B (0.49) USP2GLAKDM4EALDH1A1HSD17B10
SCHEMBL21115329 0.85 GRIN1 (0.53) USP2GLAKDM4EALDH1A1HSD17B10
SCHEMBL21115333 0.84 PDE4B (0.49) USP2GLAKDM4EALDH1A1HSD17B10
SCHEMBL21114090 0.84 HSD17B10 (0.48) USP2GLAKDM4EALDH1A1HSD17B10
SCHEMBL21113032 0.83 PDE4B (0.51) USP2GLAKDM4EALDH1A1HSD17B10
SCHEMBL21115452 0.83 KMT2A (0.54) KDM4EALDH1A1HSD17B10LMNATSHR
SCHEMBL21113771 0.82 USP2 (0.50) USP2GLAKDM4EALDH1A1HSD17B10
SCHEMBL21112855 0.82 USP2 (0.50) USP2GLAKDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3502099-B1 CYCLIC COMPOUND ACTING AS PDE4 INHIBITOR MEDSHINE DISCOVERY INC (CN) 2020-12-09 EP disclosed
EP-3502099-A1 CYCLIC COMPOUND ACTING AS PDE4 INHIBITOR Medshine Discovery Inc. (CN) 2019-06-26 EP disclosed