SCHEMBL21136716

SCHEMBL21136716

COc1cccc(F)c1-c1c(Cl)cc2c(N3CCN(C(=O)OC(C)(C)C)CC3CO)c([N+](=O)[O-])cnc2c1F

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KRAS P01116 6/20 0.41
TNF P01375 3/20 0.39
LITAF Q99732 3/20 0.39
MAP4K1 Q92918 4/20 0.38
NTRK1 P04629 2/20 0.38
BTK Q06187 1/20 0.35
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
MET P08581 2/20 0.35
MAP4K2 Q12851 2/20 0.35
STK4 Q13043 2/20 0.35
EGFR P00533 1/20 0.34
HMOX2 P30519 1/20 0.34
CRYZ Q08257 1/20 0.34
VAT1 Q99536 1/20 0.34
RTN4 Q9NQC3 1/20 0.34
GPR119 Q8TDV5 1/20 0.34
ALK Q9UM73 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21099285 1.00 KRAS (0.41) KRASTNFLITAFMAP4K1NTRK1
SCHEMBL21050970 0.91 KRAS (0.43) KRASMAP4K1NTRK1MAP4K2STK4
SCHEMBL21050961 0.91 KRAS (0.43) KRASMAP4K1NTRK1MAP4K2STK4
SCHEMBL21099404 0.90 KRAS (0.41) KRASTNFLITAFBTKCCNT1
SCHEMBL21099600 0.84 KCNH2 (0.37) BTKMETGPR119
SCHEMBL21136780 0.84 KCNH2 (0.37) BTKMETGPR119
SCHEMBL21050845 0.82 KRAS (0.45) KRASMAP4K1NTRK1EGFRHMOX2
SCHEMBL21099295 0.81 KRAS (0.37) KRASTNFLITAFMAP4K1NTRK1
SCHEMBL21099583 0.81 KRAS (0.63) KRASTNFLITAFALK
SCHEMBL21137320 0.80 KRAS (0.43) KRASTNFLITAFMAP4K1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019110751-A1 TETRACYCLIC COMPOUNDS AS INHIBITORS OF G12C MUTANT RAS PROTEIN, FOR USE AS ANTI-CANCER AGENTS ASTRAZENECA AB (SE) 2019-06-13 WO disclosed