SCHEMBL21138838

SCHEMBL21138838

O=CC(=O)N1CCC2(CC1)COc1cc(C(F)(F)F)ccc12

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 15/20 0.61
TDO2 P48775 15/20 0.61
CYP2C9 P11712 1/20 0.51
CYP3A4 P08684 1/20 0.47
S1PR5 Q9H228 4/20 0.41
S1PR1 P21453 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21138076 0.96 IDO1 (0.64) IDO1TDO2CYP2C9CYP3A4S1PR5
SCHEMBL21061068 0.83 IDO1 (0.66) IDO1TDO2CYP2C9CYP3A4S1PR5
SCHEMBL21138148 0.81 IDO1 (0.66) IDO1TDO2CYP2C9CYP3A4S1PR5
SCHEMBL21138034 0.76 IDO1 (1.00) IDO1TDO2CYP2C9CYP3A4
SCHEMBL21430773 0.76 IDO1 (0.52) IDO1TDO2CYP2C9CYP3A4
SCHEMBL21408574 0.75 IDO1 (0.52) IDO1TDO2CYP2C9CYP3A4
SCHEMBL21138413 0.75 IDO1 (0.50) IDO1TDO2CYP2C9CYP3A4
SCHEMBL12569945 0.73 GPR183 (0.49) IDO1TDO2S1PR5
Hydrochloric Acid SCHEMBL22635733 0.72 IDO1 (0.47) IDO1TDO2CYP2C9CYP3A4
SCHEMBL23271205 0.72 IDO1 (0.56) IDO1TDO2CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019115586-A1 OXALAMIDES AS MODULATORS OF INDOLEAMINE 2,3-DIOXYGENASE Phenex Discovery Verwaltungs-GmbH (DE) 2019-06-20 WO disclosed