SCHEMBL21155968

SCHEMBL21155968

C=NC(=O)C(=C)/C=C(\O)Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.42
CES2 O00748 1/20 0.42
AKR1B1 P15121 1/20 0.42
CTBP2 P56545 1/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
HIF1A Q16665 1/20 0.37
ALDH1A1 P00352 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MAPK1 P28482 1/20 0.36
EPHX2 P34913 1/20 0.36
PAM P19021 2/20 0.35
ATM Q13315 1/20 0.35
TSHR P16473 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20344509 0.79 CES1 (0.45) CES1CES2AKR1B1CTBP2MEN1
SCHEMBL19980308 0.75 CES1 (0.41) CES1CES2AKR1B1MEN1KMT2A
SCHEMBL15964742 0.68 CES1 (0.48) CES1CES2AKR1B1CTBP2MEN1
SCHEMBL19980209 0.66 CES1 (0.45) CES1CES2AKR1B1CTBP2MEN1
SCHEMBL11401352 0.65 CES1 (0.54) CES1CES2AKR1B1CTBP2MEN1
SCHEMBL162822 0.65 CES1 (0.54) CES1CES2AKR1B1CTBP2MEN1
SCHEMBL1333665 0.65 CES1 (0.52) CES1CES2AKR1B1CTBP2MEN1
Phenylacetic Acid SCHEMBL6547063 0.65 AKR1B1 (0.94) CES1CES2AKR1B1MEN1KMT2A
SCHEMBL28200225 0.64 CES1 (0.58) CES1CES2AKR1B1CTBP2MEN1
SCHEMBL41907 0.64 CES1 (0.58) CES1CES2AKR1B1CTBP2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3508484-A1 HETEROCYCLIC AMIDES AS KINASE INHIBITORS GlaxoSmithKline Intellectual Property Development Limited (GB) 2019-07-10 EP disclosed