SCHEMBL21155993

SCHEMBL21155993

CNc1cccc(-c2cccc3cnc(Nc4ccc(N5CCN(CCO)CC5)cc4)nc23)c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 3/20 0.75
JAK2 O60674 1/20 0.62
BRD4 O60885 1/20 0.62
FGFR1 P11362 3/20 0.61
KDR P35968 3/20 0.61
EGFR P00533 3/20 0.59
PTK2 Q05397 9/20 0.51
LCK P06239 1/20 0.51
FYN P06241 1/20 0.51
FES P07332 1/20 0.51
RET P07949 1/20 0.51
ROS1 P08922 1/20 0.51
CDK4 P11802 1/20 0.51
SRC P12931 1/20 0.51
JAK1 P23458 1/20 0.51
TYK2 P29597 1/20 0.51
JAK3 P52333 1/20 0.51
EPHB1 P54762 1/20 0.51
CSNK2A1 P68400 1/20 0.51
DDR1 Q08345 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19119650 0.90 FGFR2 (0.81) FGFR2JAK2BRD4FGFR1KDR
SCHEMBL29848096 0.89 FGFR2 (0.71) FGFR2JAK2BRD4FGFR1KDR
SCHEMBL16515483 0.89 FGFR2 (0.71) FGFR2JAK2BRD4FGFR1KDR
SCHEMBL20807734 0.88 FGFR1 (0.77) FGFR2JAK2BRD4FGFR1KDR
SCHEMBL16513666 0.86 FGFR2 (1.00) FGFR2JAK2BRD4FGFR1KDR
SCHEMBL20807685 0.85 EGFR (0.79) FGFR2JAK2BRD4FGFR1KDR
Maleic Acid SCHEMBL16514711 0.83 FGFR2 (0.93) FGFR2JAK2BRD4FGFR1KDR
Fumaric Acid SCHEMBL16823056 0.83 FGFR2 (0.93) FGFR2JAK2BRD4FGFR1KDR
SCHEMBL22464992 0.81 FGFR2 (0.87) FGFR2JAK2BRD4FGFR1KDR
SCHEMBL16515032 0.81 FGFR2 (0.87) FGFR2JAK2BRD4FGFR1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3508204-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Neupharma, Inc. (US) 2019-07-10 EP disclosed