SCHEMBL21158012

SCHEMBL21158012

Cn1ncc(-c2ccc(OC3CCCCC3)cn2)c1CO

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.40
SLCO1B1 Q9Y6L6 1/20 0.40
CYP4A11 Q02928 3/20 0.38
CYP4F2 P78329 2/20 0.38
BMPR1B O00238 2/20 0.36
BMPR1A P36894 2/20 0.36
ACVRL1 P37023 2/20 0.36
ACVR1 Q04771 2/20 0.36
ACACB O00763 3/20 0.36
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36
WNT1 P04628 2/20 0.35
GSK3B P49841 2/20 0.35
DYRK1A Q13627 2/20 0.35
ACVR1B P36896 1/20 0.35
FGFR1 P11362 1/20 0.35
FGFR2 P21802 1/20 0.35
FGFR4 P22455 1/20 0.35
FGFR3 P22607 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24556782 0.88 ABCB11 (0.38) ABCB11SLCO1B1CYP4A11CYP4F2BMPR1B
SCHEMBL22578295 0.85 SLCO1B1 (0.55) ABCB11SLCO1B1CYP4A11CYP4F2WNT1
SCHEMBL22463678 0.85 SLCO1B1 (0.55) ABCB11SLCO1B1CYP4A11CYP4F2WNT1
SCHEMBL22578294 0.85 SLCO1B1 (0.55) ABCB11SLCO1B1CYP4A11CYP4F2WNT1
SCHEMBL22576690 0.81 SLCO1B1 (0.45) ABCB11SLCO1B1CYP4A11CYP4F2ACACB
SCHEMBL22577733 0.81 SLCO1B1 (0.45) ABCB11SLCO1B1CYP4A11CYP4F2ACACB
SCHEMBL31212636 0.81 SLCO1B1 (0.45) ABCB11SLCO1B1CYP4A11CYP4F2ACACB
SCHEMBL21157294 0.80 NPC1 (0.39) ABCB11SLCO1B1CYP4A11CYP4F2BMPR1B
SCHEMBL30338659 0.80 SLCO1B1 (0.62) ABCB11SLCO1B1CYP4A11CYP4F2LPAR1
SCHEMBL21156725 0.80 LPAR1 (0.37) ABCB11SLCO1B1WNT1GSK3BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3728216-B1 PYRAZOLE N-LINKED CARBAMOYL CYCLOHEXYL ACIDS AS LPA ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2023-09-06 EP disclosed
EP-3727589-B1 CYCLOHEXYL ACID PYRAZOLE AZOLES AS LPA ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2022-06-29 EP disclosed
WO-2019126085-A1 PYRAZOLE N-LINKED CARBAMOYL CYCLOHEXYL ACIDS AS LPA ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2019-06-27 WO disclosed