SCHEMBL21158804

SCHEMBL21158804

CCCC(=O)N(C)N(C)C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PHF8 Q9UPP1 1/20 0.61
KDM2A Q9Y2K7 1/20 0.61
ALDH1A1 P00352 4/20 0.44
CES2 O00748 3/20 0.43
CES1 P23141 3/20 0.43
HDAC3 O15379 4/20 0.41
HDAC1 Q13547 4/20 0.41
HDAC2 Q92769 4/20 0.41
HDAC8 Q9BY41 4/20 0.41
FFAR3 O14843 3/20 0.41
TSHR P16473 2/20 0.39
TP53 P04637 1/20 0.38
HDAC6 Q9UBN7 1/20 0.36
JAK2 O60674 1/20 0.35
S1PR4 O95977 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8847986 0.81 ALDH1A1 (0.42) PHF8KDM2AALDH1A1CES2CES1
SCHEMBL3263226 0.78 PHF8 (0.61) PHF8KDM2AALDH1A1HDAC3HDAC1
SCHEMBL2387300 0.78 ALDH1A1 (0.44) PHF8KDM2AALDH1A1CES2CES1
SCHEMBL3260392 0.77 PHF8 (0.48) PHF8KDM2AALDH1A1CTSD
SCHEMBL14032784 0.77 ALDH1A1 (0.48) PHF8KDM2AALDH1A1CES2CES1
SCHEMBL139743 0.77
SCHEMBL4774587 0.77
SCHEMBL1801852 0.76 ALDH1A1 (0.42) PHF8KDM2AALDH1A1CES2CES1
Hydrochloric Acid SCHEMBL8373771 0.74 ALDH1A1 (0.67) ALDH1A1CES2CES1HDAC3HDAC1
Bromide SCHEMBL8373855 0.74 ALDH1A1 (0.67) ALDH1A1CES2CES1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3737665-A1 PRODRUGS OF KETAMINE, COMPOSITIONS AND USES THEREOF XW Laboratories Inc. (KY) 2020-11-18 EP disclosed
WO-2019137381-A1 PRODRUGS OF KETAMINE, COMPOSITIONS AND USES THEREOF XW LABORATORIES, INC. (CN) 2019-07-18 WO disclosed