SCHEMBL21167657

SCHEMBL21167657

Cc1cc(Nc2cnc(N)c(NCc3ccc4ncccc4c3)n2)cc(C)n1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.41
DHFR P00374 1/20 0.41
KDR P35968 7/20 0.39
MET P08581 2/20 0.39
HDAC6 Q9UBN7 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
TERT O14746 2/20 0.37
KLKB1 P03952 1/20 0.37
KLK1 P06870 1/20 0.37
SYK P43405 1/20 0.37
HDAC3 O15379 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21167575 0.92 NPC1 (0.41) NPC1ABCB1ABCC1ABCG2DHFR
SCHEMBL21167454 0.91 NPC1 (0.44) NPC1ABCB1ABCC1ABCG2DHFR
SCHEMBL21167629 0.88 NPC1 (0.44) NPC1DHFRKDRMETHDAC6
SCHEMBL21167437 0.87 PIK3CA (0.42) NPC1ABCB1ABCC1ABCG2DHFR
SCHEMBL21167728 0.87 NPC1 (0.43) NPC1DHFRKDRMETHDAC6
SCHEMBL21167462 0.87 KDR (0.42) NPC1DHFRKDRMETHDAC6
SCHEMBL21167592 0.86 NPC1 (0.42) NPC1DHFRKDRMETHDAC6
SCHEMBL21167366 0.85 NPC1 (0.43) NPC1DHFRKDRMETHDAC6
SCHEMBL21167621 0.85 NPC1 (0.40) NPC1ABCB1ABCC1ABCG2DHFR
SCHEMBL29314302 0.85 NPC1 (0.43) NPC1ABCB1ABCC1ABCG2DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3795573-B1 CERTAIN TRIAZOLOPYRAZINES, COMPOSITIONS THEREOF AND METHODS OF USE THEREFOR HUTCHISON MEDIPHARMA LTD (CN) 2022-07-06 EP disclosed
EP-3795573-A1 CERTAIN TRIAZOLOPYRIDINES AND TRIAZOLOPYRIDINES, COMPOSITIONS THEREOF AND METHODS OF USE THEREFOR Hutchison Medipharma Limited (CN) 2021-03-24 EP disclosed
EP-3511330-B1 SYNTHETIC INTERMEDIATE USEFUL IN THE PREPARATION OF TRIAZOLOPYRIDINE C-MET INHIBITORS HUTCHISON MEDIPHARMA LTD (CN) 2020-09-30 EP disclosed
EP-3511330-A1 SYNTHETIC INTERMEDIATE USEFUL IN THE PREPARATION OF TRIAZOLOPYRIDINE C-MET INHIBITORS Hutchison Medipharma Limited (CN) 2019-07-17 EP disclosed