SCHEMBL21167672

SCHEMBL21167672

Cn1cc(-c2cnc(N)c(NCc3cc(N)c(C=N)s3)n2)cn1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 7/20 0.56
MAPK1 P28482 3/20 0.37
AURKA O14965 3/20 0.35
AURKB Q96GD4 3/20 0.35
FGFR3 P22607 4/20 0.35
FGFR1 P11362 3/20 0.35
FGFR2 P21802 3/20 0.35
MAP4K1 Q92918 2/20 0.35
KDR P35968 1/20 0.34
LDHA P00338 1/20 0.34
LDHB P07195 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22475817 0.90 CSF1R (0.45) CSF1RMAPK1AURKBFGFR3FGFR1
SCHEMBL21167614 0.87 CSF1R (0.42) CSF1RMAPK1AURKBMAP4K1
SCHEMBL21167411 0.87 CSF1R (0.41) CSF1RFGFR3FGFR1FGFR2KDR
SCHEMBL21167440 0.86 CSF1R (0.42) CSF1RFGFR3FGFR1FGFR2KDR
SCHEMBL24591027 0.84 CSF1R (0.39) CSF1RFGFR3FGFR1FGFR2LDHA
SCHEMBL21167328 0.81 MAPK1 (0.36) CSF1RMAPK1AURKBFGFR2LDHA
SCHEMBL24591047 0.80 CSF1R (0.37) CSF1RMAPK1AURKAAURKBFGFR3
SCHEMBL22475672 0.79 CSF1R (0.41) CSF1RMAPK1FGFR3FGFR1FGFR2
SCHEMBL22475803 0.78 SYK (0.35) CSF1RFGFR3FGFR1FGFR2KDR
SCHEMBL24591126 0.78 LRRK2 (0.36) CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3511330-A1 SYNTHETIC INTERMEDIATE USEFUL IN THE PREPARATION OF TRIAZOLOPYRIDINE C-MET INHIBITORS Hutchison Medipharma Limited (CN) 2019-07-17 EP disclosed