SCHEMBL21167733

SCHEMBL21167733

NNc1ccc(Nc2cccnc2)nc1NCc1ccc2ncccc2c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
SYK P43405 2/20 0.40
KDR P35968 6/20 0.39
HDAC6 Q9UBN7 1/20 0.38
FLT1 P17948 1/20 0.36
RAB9A P51151 2/20 0.36
HDAC3 O15379 1/20 0.36
CSF1R P07333 1/20 0.36
SSTR3 P32745 1/20 0.35
KDM4E B2RXH2 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
BACE1 P56817 1/20 0.35
PIK3CA P42336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22475819 0.90 NPC1 (0.43) NPC1SYKKDRHDAC6FLT1
SCHEMBL21167731 0.88 NPC1 (0.43) NPC1SYKKDRHDAC6RAB9A
SCHEMBL22475714 0.86 BACE1 (0.41) NPC1SYKKDRRAB9ABACE1
SCHEMBL21167728 0.84 NPC1 (0.43) NPC1SYKKDRHDAC6RAB9A
SCHEMBL22475999 0.82 IGF1R (0.41) NPC1SYKKDRHDAC6
SCHEMBL22475673 0.82 KDR (0.40) NPC1SYKKDRHDAC6FLT1
SCHEMBL21167726 0.81 SYK (0.40) NPC1SYKKDRHDAC6BACE1
SCHEMBL22475963 0.79 KDR (0.43) NPC1SYKKDR
SCHEMBL21167658 0.77 NPC1 (0.45) NPC1SYKKDRHDAC6FLT1
SCHEMBL24591152 0.76 NPC1 (0.43) NPC1SYKKDRHDAC6FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3511330-A1 SYNTHETIC INTERMEDIATE USEFUL IN THE PREPARATION OF TRIAZOLOPYRIDINE C-MET INHIBITORS Hutchison Medipharma Limited (CN) 2019-07-17 EP disclosed