SCHEMBL21170249

SCHEMBL21170249

C=C(N)c1cc(-c2ccc(NCC(C)(C)c3ncccc3F)nn2)ccc1N

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IL1B P01584 10/20 0.33
CDC7 O00311 1/20 0.32
DAPK3 O43293 1/20 0.32
ROCK2 O75116 1/20 0.32
PRKD3 O94806 1/20 0.32
MAP4K4 O95819 1/20 0.32
PAK4 O96013 1/20 0.32
PIM1 P11309 1/20 0.32
PRKACA P17612 1/20 0.32
CDK2 P24941 1/20 0.32
FLT3 P36888 1/20 0.32
CSNK1A1 P48729 1/20 0.32
CDK8 P49336 1/20 0.32
CLK2 P49760 1/20 0.32
GSK3B P49841 1/20 0.32
CDK7 P50613 1/20 0.32
CDK9 P50750 1/20 0.32
PRKX P51817 1/20 0.32
JAK3 P52333 1/20 0.32
CDK5 Q00535 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21170329 0.86 IL1B (0.34) IL1BCDC7DAPK3ROCK2PRKD3
SCHEMBL21170097 0.84 CDC7 (0.33) IL1BCDC7DAPK3ROCK2PRKD3
SCHEMBL21170213 0.83 IL1B (0.37) IL1BTNF
SCHEMBL21170327 0.81 IL1B (0.33) IL1BTNF
SCHEMBL12286826 0.80 PDE4A (0.38)
SCHEMBL21170344 0.80 IL1B (0.37) IL1BTNF
SCHEMBL21170111 0.80 IL1B (0.33) IL1BTNF
SCHEMBL21170275 0.79 IL1B (0.34) IL1BTNF
SCHEMBL21170497 0.79 IL1B (0.36) IL1BTNF
SCHEMBL12287071 0.79 PDPK1 (0.45) CDK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3127541-B1 CERTAIN AMINO-PYRIDAZINES, COMPOSITIONS THEREOF, AND METHODS OF THEIR USE CYTOKINETICS INC (US) 2019-07-17 EP disclosed