SCHEMBL21173305

SCHEMBL21173305

CCOC(=O)[C@@H]1[C@H]2CC[C@H](C2)N1C(O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PREP P48147 1/20 0.36
CTSL P07711 1/20 0.34
KCNH2 Q12809 1/20 0.33
MEN1 O00255 2/20 0.32
ALDH1A1 P00352 2/20 0.32
KMT2A Q03164 2/20 0.32
TSHR P16473 1/20 0.32
MAPT P10636 1/20 0.32
FKBP1A P62942 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21173306 0.82 PREP (0.39) PREP
SCHEMBL15934593 0.74 PREP (0.61) PREPCTSLMEN1ALDH1A1KMT2A
SCHEMBL2097353 0.74 PREP (0.61) PREPCTSLMEN1ALDH1A1KMT2A
SCHEMBL6621402 0.74 PREP (0.61) PREPCTSLMEN1ALDH1A1KMT2A
SCHEMBL6620964 0.74 PREP (0.61) PREPCTSLMEN1ALDH1A1KMT2A
SCHEMBL15934580 0.74 PREP (0.61) PREPCTSLMEN1ALDH1A1KMT2A
SCHEMBL17862217 0.74 PREP (0.61) PREPCTSLMEN1ALDH1A1KMT2A
SCHEMBL12294933 0.74 PREP (0.61) PREPCTSLMEN1ALDH1A1KMT2A
SCHEMBL14583166 0.74 PREP (0.37) PREP
SCHEMBL4736905 0.72 MAPT (0.36) KCNH2MEN1ALDH1A1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3191487-B1 SPIROCYCLIC INHIBITORS OF CATHEPSIN C BOEHRINGER INGELHEIM INT (DE) 2019-08-07 EP disclosed
EP-3511331-A1 SPIROCYCLIC INHIBITORS OF CATHEPSIN C Boehringer Ingelheim International GmbH (DE) 2019-07-17 EP disclosed